SCHEMBL7497802

SCHEMBL7497802

COC(=O)CC[C@H](NC(=O)c1cc(CCC2CNc3nc(N)nc(O)c3C2)c[nH]1)C(=O)OC

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GART P22102 5/20 0.43
DHFR P00374 3/20 0.40
ALDH1A1 P00352 1/20 0.32
MAPK1 P28482 1/20 0.32
ALOX5 P09917 1/20 0.32
ATIC P31939 3/20 0.32
KDR P35968 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7495297 0.87 GART (0.57) GARTDHFRATIC
SCHEMBL7496547 0.86 GART (0.43) GARTDHFRALOX5ATICKDR
SCHEMBL7497455 0.85 GART (0.43) GARTDHFRALDH1A1MAPK1ALOX5
SCHEMBL7497451 0.85 GART (0.43) GARTDHFRALDH1A1MAPK1ALOX5
SCHEMBL8017846 0.84 GART (0.40) GARTDHFRALDH1A1MAPK1KDR
SCHEMBL8017849 0.84 GART (0.40) GARTDHFRALDH1A1MAPK1KDR
SCHEMBL7503308 0.80 GART (0.58) GARTDHFRATIC
SCHEMBL7493397 0.79 DHFR (0.43) GARTDHFR
SCHEMBL9383614 0.78 GART (0.56) GARTDHFRALDH1A1ATIC
SCHEMBL9383606 0.78 GART (0.56) GARTDHFRALDH1A1ATIC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0904271-A4 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES UNIV PRINCETON (US) 2002-01-23 EP disclosed
US-6066639-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2000-05-23 US disclosed
EP-0904271-A1 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1999-03-31 EP disclosed
WO-1997041115-A1 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1997-11-06 WO disclosed