SCHEMBL7498302

SCHEMBL7498302

COc1cccc(-c2cc3c(O)ncnc3[nH]2)c1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 1/20 0.59
GSK3B P49841 2/20 0.56
CCNB2 O95067 1/20 0.56
CDK1 P06493 1/20 0.56
CCNB1 P14635 1/20 0.56
GSK3A P49840 1/20 0.56
CDK5 Q00535 1/20 0.56
CDK5R1 Q15078 1/20 0.56
CCNB3 Q8WWL7 1/20 0.56
MAPKAPK2 P49137 1/20 0.53
EIF2AK2 P19525 1/20 0.52
KIT P10721 2/20 0.49
IKBKB O14920 1/20 0.48
CHUK O15111 1/20 0.48
MAP4K4 O95819 1/20 0.46
EGFR P00533 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4903666 0.85 EGFR (0.57) CSF1RGSK3BCCNB2CDK1CCNB1
SCHEMBL7495582 0.84 CSF1R (0.59) CSF1RGSK3BCCNB2CDK1CCNB1
SCHEMBL1897594 0.80 EGFR (0.55) CSF1RKITEGFR
SCHEMBL30588943 0.80 EGFR (0.55) CSF1RKITEGFR
SCHEMBL8089650 0.78 CCNT1 (0.47) CSF1RCHUKEGFR
SCHEMBL27444977 0.77 EGFR (0.55) CSF1RKITEGFR
SCHEMBL7497561 0.77 RIPK1 (0.49) CSF1RGSK3BEIF2AK2KITEGFR
SCHEMBL2444894 0.76 CCNB2 (0.64) CSF1RGSK3BCCNB2CDK1CCNB1
SCHEMBL2461351 0.76 EGFR (0.57) CSF1RCDK1MAP4K4EGFR
SCHEMBL7504170 0.75 CSF1R (0.54) CSF1REGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836605-B1 PYRROLOPYRIMIDINES AND PROCESSES FOR THE PREPARATION THEREOF NOVARTIS AG (CH) 2002-02-06 EP disclosed
US-6140332-A Pyrrolopyrimidines and processes for the preparation thereof NOVARTIS AG (CH) 2000-10-31 US disclosed
US-6096749-A ANTITUMOR, EPIDERMAL GROWTH FACTOR NOVARTIS CORPORATION (US) 2000-08-01 US disclosed
EP-0836605-A1 PYRROLOPYRIMIDINES AND PROCESSES FOR THE PREPARATION THEREOF Novartis AG (CH) 1998-04-22 EP disclosed
WO-1997002266-A1 PYRROLOPYRIMIDINES AND PROCESSES FOR THE PREPARATION THEREOF NOVARTIS AG (CH) 1997-01-23 WO disclosed
EP-0682027-A1 Pyrrolopyrimidine derivatives with antiproliferative action CIBA-GEIGY AG (CH) 1995-11-15 EP disclosed