SCHEMBL7498558

SCHEMBL7498558

Nc1nc(O)c2c(n1)NCC(CCc1cc(C(=O)O)c[nH]1)C2

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.41
GART P22102 3/20 0.36
NOS1 P29475 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7502010 0.83 HCAR2 (0.42) DHFR
SCHEMBL7490675 0.83 DHFR (0.56) DHFRGARTNOS1
SCHEMBL8874134 0.83 DHFR (0.56) DHFRGARTNOS1
SCHEMBL7491867 0.83 GART (0.57) DHFRGART
Hydrochloric Acid SCHEMBL7487428 0.82 DHFR (0.55) DHFRGARTNOS1
Hydrochloric Acid SCHEMBL8875657 0.82 DHFR (0.55) DHFRGARTNOS1
SCHEMBL7493397 0.82 DHFR (0.43) DHFRGARTNOS1
SCHEMBL7494746 0.80 DHFR (0.42) DHFRGARTNOS1
SCHEMBL7496547 0.79 GART (0.43) DHFRGART
SCHEMBL7487410 0.76 DHFR (0.57) DHFRGARTNOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0904271-A4 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES UNIV PRINCETON (US) 2002-01-23 EP disclosed
US-6066639-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2000-05-23 US disclosed
EP-0904271-A1 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1999-03-31 EP disclosed
WO-1997041115-A1 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1997-11-06 WO disclosed