SCHEMBL7502010

SCHEMBL7502010

Nc1nc(O)c2c(n1)NCC(CCc1cc(C(=O)O)n[nH]1)C2

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 11/20 0.42
HCAR3 P49019 2/20 0.41
DHFR P00374 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7499714 0.83 GART (0.54) DHFR
SCHEMBL8018583 0.83 GART (0.54) DHFR
SCHEMBL7498558 0.83 DHFR (0.41) DHFR
SCHEMBL7494746 0.82 DHFR (0.42) DHFR
SCHEMBL7490675 0.81 DHFR (0.56) DHFR
SCHEMBL8874134 0.81 DHFR (0.56) DHFR
SCHEMBL8017846 0.80 GART (0.40) HCAR2DHFR
SCHEMBL8017849 0.80 GART (0.40) HCAR2DHFR
Hydrochloric Acid SCHEMBL8875657 0.80 DHFR (0.55) DHFR
Hydrochloric Acid SCHEMBL7487428 0.80 DHFR (0.55) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0904271-A4 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES UNIV PRINCETON (US) 2002-01-23 EP disclosed
US-6066639-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2000-05-23 US disclosed
EP-0904271-A1 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1999-03-31 EP disclosed
WO-1997041115-A1 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1997-11-06 WO disclosed