SCHEMBL7499006

SCHEMBL7499006

CC(=O)N[C@H](C(=O)c1noc(Cc2cccc(C(F)(F)F)c2)n1)C(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.48
NPC1 O15118 2/20 0.48
PRSS1 P07477 3/20 0.46
PRSS2 P07478 3/20 0.46
PRSS3 P35030 3/20 0.46
TPSAB1 Q15661 3/20 0.46
KMT2A Q03164 6/20 0.44
HTT P42858 1/20 0.44
ZAP70 P43403 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 4/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
POLB P06746 1/20 0.39
EPHX1 P07099 1/20 0.39
CSGALNACT1 Q8TDX6 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8165421 0.83 KMT2A (0.43) RAB9ANPC1PRSS1PRSS2PRSS3
SCHEMBL8491074 0.80 PRSS1 (0.43) RAB9ANPC1PRSS1PRSS2PRSS3
SCHEMBL7505093 0.80 PRSS1 (0.41) RAB9ANPC1PRSS1PRSS2PRSS3
SCHEMBL892526 0.79 KMT2A (0.47) RAB9ANPC1PRSS1PRSS2PRSS3
SCHEMBL8491451 0.77 ELANE (0.64)
SCHEMBL8495148 0.77 PRSS1 (0.40) RAB9ANPC1PRSS1PRSS2PRSS3
SCHEMBL7208823 0.77 PRSS1 (0.40) RAB9ANPC1PRSS1PRSS2PRSS3
SCHEMBL893046 0.75 KMT2A (0.56) RAB9ANPC1PRSS1PRSS2PRSS3
SCHEMBL8436306 0.70 PRSS1 (0.51) RAB9ANPC1PRSS1PRSS2PRSS3
SCHEMBL1114503 0.70 MEN1 (0.59) KMT2AHTTSMN1; SMN2MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0954526-A2 SERINE PROTEASE INHIBITORS CORTECH, INC. (US) 1999-11-10 EP disclosed
WO-1998024806-A2 SUBSTITUTED OXADIAZOLE, THIADIAZOLE AND TRIAZOLE SERINE PROTEASE INHIBITORS CORTECH, INC. (US) 1998-06-11 WO disclosed