SCHEMBL7499299

SCHEMBL7499299

CCCCCCCCOc1cc(C(=O)OC)ccc1N

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.60
CYP2D6 P10635 1/20 0.60
TSHR P16473 1/20 0.60
SLC6A2 P23975 1/20 0.60
SCN1A P35498 1/20 0.60
SLC6A3 Q01959 1/20 0.60
KCNH2 Q12809 1/20 0.60
HIF1A Q16665 1/20 0.60
SCN2A Q99250 1/20 0.60
SCN3A Q9NY46 1/20 0.60
HRH3 Q9Y5N1 1/20 0.60
RAD52 P43351 1/20 0.59
SMPD1 P17405 6/20 0.55
MGLL Q99685 2/20 0.52
ERAP2 Q6P179 1/20 0.51
LNPEP Q9UIQ6 1/20 0.51
ALDH1A1 P00352 2/20 0.50
NPC1 O15118 1/20 0.50
MAPT P10636 1/20 0.50
RAB9A P51151 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL222268 0.94 CYP1A2 (0.67) CYP1A2CYP2D6TSHRSLC6A2SCN1A
SCHEMBL11949139 0.90 CYP1A2 (0.57) CYP1A2CYP2D6TSHRSLC6A2SCN1A
SCHEMBL11600843 0.89 SMPD1 (0.55) CYP1A2CYP2D6SCN1AKCNH2SCN2A
SCHEMBL8085916 0.87 CYP1A2 (0.73) CYP1A2CYP2D6TSHRSLC6A2SCN1A
SCHEMBL24950547 0.87 SMPD1 (0.67) SMPD1MGLLALDH1A1HPGDTHRA
SCHEMBL9565566 0.87 SMPD1 (0.67) SMPD1MGLLALDH1A1HPGDTHRA
SCHEMBL967401 0.87 SMPD1 (0.67) SMPD1MGLLALDH1A1HPGDTHRA
SCHEMBL9304902 0.87 SMPD1 (0.67) SMPD1MGLLALDH1A1HPGDTHRA
SCHEMBL7335792 0.85 SMPD1 (0.64) SMPD1MGLLALDH1A1HPGDTHRA
SCHEMBL8085032 0.85 ALDH1A1 (0.62) CYP1A2CYP2D6TSHRSLC6A2SCN1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1124788-A4 BIS(HALOETHYL)AMINOBENZENE DERIVATIVES SHIONOGI BIORES CORP (US) 2002-11-06 EP disclosed
US-6433199-B1 ANTITUMOR, ANTICANCER AGENTS SHIONOGI BIORESEARCH CORPORATION 2002-08-13 US disclosed
EP-1124788-A2 BIS(HALOETHYL)AMINOBENZENE DERIVATIVES Shionogi Bioresearch Corporation (US) 2001-08-22 EP disclosed
US-6137003-A Bis (haloethyl) aminobenzene derivatives SHIONOGI BIORESEARCH (US) 2000-10-24 US disclosed
WO-2000024361-A2 BIS(HALOETHYL)AMINOBENZENE DERIVATIVES SHIONOGI BIORESEARCH CORP. (US) 2000-05-04 WO disclosed
US-5969133-A Bioreductive cytotoxic agents SHIONGI BIORESEARCH CORP. (US) 1999-10-19 US disclosed