SCHEMBL7500218

SCHEMBL7500218

Cn1[nH]c(=O)c2c1NC1=C(C(=O)CC1)C2c1ccc(Cl)c([N+](=O)[O-])c1.O=Cc1ccc(Cl)c([N+](=O)[O-])c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 1/20 0.43
ABCC9 O60706 6/20 0.42
ABCC8 Q09428 6/20 0.42
KCNJ11 Q14654 6/20 0.42
KCNJ8 Q15842 6/20 0.42
BRD4 O60885 1/20 0.38
BRDT Q58F21 1/20 0.38
MAPT P10636 7/20 0.33
MAPK1 P28482 2/20 0.33
RAB9A P51151 1/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C19 P33261 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
ALDH1A1 P00352 2/20 0.32
LMNA P02545 1/20 0.32
KMT2A Q03164 1/20 0.32
PKM P14618 1/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
RECQL P46063 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6641885 0.93 ABCC9 (0.47) VCAM1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL6643734 0.81 BRD4 (0.47) ABCC9ABCC8KCNJ11KCNJ8BRD4
SCHEMBL6643320 0.79 ABCC9 (0.38) VCAM1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL7548646 0.78 ABCC9 (0.44) ABCC9ABCC8KCNJ11KCNJ8BRD4
SCHEMBL6649861 0.78 ABCC9 (0.48) VCAM1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL7499328 0.78 ABCC9 (0.43) ABCC9ABCC8KCNJ11KCNJ8BRD4
SCHEMBL6856477 0.77 ABCC9 (0.42) VCAM1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL6928832 0.77 ABCC9 (0.54) ABCC9ABCC8KCNJ11KCNJ8MAPT
SCHEMBL6643759 0.76 ABCC9 (0.45) ABCC9ABCC8KCNJ11KCNJ8BRD4
SCHEMBL6644997 0.73 ABCC9 (0.49) ABCC9ABCC8KCNJ11KCNJ8BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1259510-A2 TRICYCLIC DIHYDROPYRAZOLONE AND TRICYCLIC DIHYDROISOXAZOLONE POTASSIUM CHANNEL OPENERS ABBOTT LABORATORIES (US) 2002-11-27 EP disclosed
WO-2001066544-A2 TRICYCLIC DIHYDROPYRAZOLONE AND TRICYCLIC DIHYDROISOXAZOLONE POTASSIUM CHANNEL OPENERS ABBOTT LABORATORIES (US) 2001-09-13 WO disclosed