SCHEMBL7500511

SCHEMBL7500511

O=C1C(Cc2ccccc2)C(c2ccccc2)=Nc2ccccc2N1Cc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.56
MAPT P10636 1/20 0.56
EP300 Q09472 1/20 0.54
CES2 O00748 13/20 0.51
POLB P06746 1/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 2/20 0.42
MAPK1 P28482 1/20 0.42
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7503888 0.83 EP300 (0.55) ALDH1A1MAPTEP300CES2POLB
SCHEMBL7499159 0.80 EP300 (0.51) ALDH1A1MAPTEP300CES2POLB
SCHEMBL7492974 0.78 EP300 (0.49) ALDH1A1MAPTEP300POLBGAA
SCHEMBL7492969 0.78 EP300 (0.49) ALDH1A1MAPTEP300POLBGAA
SCHEMBL9654418 0.76 CES2 (0.50) ALDH1A1MAPTCES2KMT2AMAPK1
SCHEMBL7507531 0.76 EP300 (0.46) ALDH1A1MAPTEP300CES2POLB
SCHEMBL29045024 0.72 CES2 (0.48) ALDH1A1MAPTEP300CES2GAA
SCHEMBL17070924 0.72 EP300 (0.62) ALDH1A1MAPTEP300CES2POLB
SCHEMBL7505364 0.72 ALDH1A1 (1.00) ALDH1A1MAPTPOLBKMT2AMAPK1
SCHEMBL7499535 0.72 ALDH1A1 (0.44) ALDH1A1MAPTEP300CES2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757681-B1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-09-18 EP disclosed
US-5834463-A CONTROLLING FERTILITY, MENSTRUAL CYCLES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-11-10 US disclosed
EP-0757681-A1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 1997-02-12 EP disclosed
WO-1995029900-A1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-11-09 WO disclosed