SCHEMBL7501562

SCHEMBL7501562

O=C1[C@H]2CCC[C@H]2N(C(=O)CBr)c2ccccc2N1CCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CASR P41180 2/20 0.46
ALDH1A1 P00352 8/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
CCKBR P32239 1/20 0.41
XIAP P98170 4/20 0.40
ALOX12 P18054 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
ALDH2 P05091 1/20 0.40
ALDH3A1 P30838 1/20 0.40
PARK7 Q99497 1/20 0.40
CYP3A4 P08684 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7499726 0.94 ALDH1A1 (0.42) CASRALDH1A1KDM4ELMNAXIAP
SCHEMBL7500262 0.89 ALDH1A1 (0.52) ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL7495825 0.89 ALDH1A1 (0.52) ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL7500658 0.86 CASR (0.48) CASRALDH1A1KDM4ELMNAXIAP
SCHEMBL7502331 0.81 ALDH1A1 (0.42) ALDH1A1LMNAMEN1KMT2A
SCHEMBL7507580 0.80 ALDH1A1 (0.45) CASRALDH1A1KDM4EXIAPALDH2
SCHEMBL7508401 0.79 ALDH1A1 (0.46) ALDH1A1ALDH2ALDH3A1SMN1; SMN2MEN1
SCHEMBL7507845 0.78 TSHR (0.43) ALDH1A1LMNASMN1; SMN2KMT2A
SCHEMBL7497359 0.78 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL7497354 0.78 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757681-B1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-09-18 EP disclosed
WO-1995029900-A1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-11-09 WO disclosed