SCHEMBL7499726

SCHEMBL7499726

O=C1[C@H]2CCC[C@H]2N(C(=O)CBr)c2ccccc2N1CCCc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
ALDH2 P05091 1/20 0.42
PKM P14618 1/20 0.42
ALDH3A1 P30838 1/20 0.42
XIAP P98170 1/20 0.41
CASR P41180 2/20 0.40
GSK3A P49840 1/20 0.39
GSK3B P49841 1/20 0.39
CHRNB4 P30926 3/20 0.38
CHRNA3 P32297 3/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
SIGMAR1 Q99720 1/20 0.37
CHRM3 P20309 1/20 0.37
KDM4E B2RXH2 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LMNA P02545 1/20 0.36
BLM P54132 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7501562 0.94 CASR (0.46) ALDH1A1ALDH2PKMALDH3A1XIAP
SCHEMBL7495825 0.87 ALDH1A1 (0.52) ALDH1A1
SCHEMBL7500262 0.87 ALDH1A1 (0.52) ALDH1A1
SCHEMBL7507580 0.87 ALDH1A1 (0.45) ALDH1A1ALDH2PKMALDH3A1XIAP
SCHEMBL7500658 0.80 CASR (0.48) ALDH1A1ALDH2ALDH3A1XIAPCASR
SCHEMBL7502331 0.79 ALDH1A1 (0.42) ALDH1A1GSK3BL3MBTL1LMNA
SCHEMBL9117259 0.78 ALDH1A1 (0.47) ALDH1A1XIAP
SCHEMBL9117256 0.78 ALDH1A1 (0.47) ALDH1A1XIAP
SCHEMBL7498239 0.78 ALDH1A1 (0.52) ALDH1A1
SCHEMBL7501263 0.78 ALDH1A1 (0.52) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757681-B1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-09-18 EP disclosed
WO-1995029900-A1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-11-09 WO disclosed