SCHEMBL750158

SCHEMBL750158

FC(F)(F)c1nnc2ccc(Cl)nn12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 1.00
KDM4E B2RXH2 2/20 0.77
SMN1; SMN2 Q16637 2/20 0.77
HTT P42858 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
CYP1A2 P05177 4/20 0.51
SCN5A Q14524 1/20 0.51
ALOX15 P16050 1/20 0.51
MAPT P10636 2/20 0.49
HPGD P15428 1/20 0.49
DYRK1A Q13627 1/20 0.49
DYRK2 Q92630 1/20 0.49
AR P10275 1/20 0.46
KCNH2 Q12809 1/20 0.46
TP53 P04637 1/20 0.46
HSD17B10 Q99714 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
XBP1 P17861 1/20 0.46
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2265102 0.87 KDM4E (1.00) ALDH1A1KDM4ESMN1; SMN2HTTTDP1
SCHEMBL2267586 0.86 ALDH1A1 (0.75) ALDH1A1KDM4ESMN1; SMN2HTTTDP1
SCHEMBL22744857 0.86 ALDH1A1 (0.75) ALDH1A1KDM4ESMN1; SMN2HTTTDP1
SCHEMBL20203879 0.86 ALDH1A1 (0.75) ALDH1A1KDM4ESMN1; SMN2HTTTDP1
SCHEMBL24616729 0.82 ALDH1A1 (0.69) ALDH1A1KDM4ESMN1; SMN2HTTTDP1
SCHEMBL2268505 0.82 ALDH1A1 (0.69) ALDH1A1KDM4ESMN1; SMN2HTTTDP1
SCHEMBL6631672 0.81 ALDH1A1 (0.69) ALDH1A1KDM4ESMN1; SMN2HTTTDP1
SCHEMBL939060 0.78 ALDH1A1 (0.64) ALDH1A1KDM4ESMN1; SMN2HTTTDP1
SCHEMBL12911394 0.78 ALDH1A1 (0.64) ALDH1A1KDM4ESMN1; SMN2HTTTDP1
SCHEMBL2362190 0.78 ALDH1A1 (0.64) ALDH1A1KDM4ESMN1; SMN2HTTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 119 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116885-A1 ION CHANNEL MODULATORS PRAXIS PREC MEDICINES INC (US) 2026-04-30 US disclosed
US-12522595-B2 Bicyclic ether O-glycoprotein-2-acetamido-2-deoxy-3-D-glucopyranosidase inhibitors BIOGEN MA INC. (US) 2026-01-13 US disclosed
US-12344615-B2 Substituted pyridines as ion channel modulators PRAXIS PRECISION MEDICINES, INC. (US) 2025-07-01 US disclosed
US-20250163068-A1 COMPOUNDS AND THEIR METHODS OF USE PRAXIS PRECISION MEDICINES, INC. 2025-05-22 US disclosed
US-20250115569-A1 SULFONAMIDE COMPOUNDS FOR THE TREATMENT OF NEUROLOGICAL CONDITIONS LARIO THERAPEUTICS LTD (GB) 2025-04-10 US disclosed
US-12152035-B2 Androgen receptor binding molecule and use thereof INDUSTRIAL TECHNOLOGY RESEARCH INSTITUTE (TW) 2024-11-26 US disclosed
WO-2024229221-A1 ANDROGEN RECEPTOR MODULATORS AND METHODS FOR THEIR USE CAPULUS THERAPEUTICS, LLC (US) 2024-11-07 WO disclosed
CN-114685601-B Androgen receptor binding molecules and uses thereof 财团法人工业技术研究院 2024-10-18 CN disclosed
EP-4397308-A2 COMPOUNDS AND THEIR METHODS OFUSE Praxis Precision Medicines, Inc. (US) 2024-07-10 EP disclosed
CN-118317950-A Sulfonamide compounds for the treatment of neurological disorders 拉里奥治疗有限公司 2024-07-09 CN disclosed
WO-2010131022-A1 [1,2,4] TRIAZOLO [4,3-B] PYRIDAZINES AS LIGANDS OF THE ANDROGEN RECEPTOR ASTRAZENECA AB (SE) 2010-11-18 WO disclosed
US-20100267699-A1 CHEMICAL COMPOUNDS - 643 ASTRAZENECA R&D 2010-10-21 US disclosed
EP-2235010-A1 BICYCLIC DERIVATIVES FOR USE IN THE TREATMENT OF ANDROGEN RECEPTOR ASSOCIATED CONDITIONS AstraZeneca AB (SE) 2010-10-06 EP disclosed
WO-2010092371-A1 TRIAZOLO [4,3-B] PYRIDAZINE DERIVATIVES AND THEIR USES FOR PROSTATE CANCER ASTRAZENECA AB (SE) 2010-08-19 WO disclosed
US-20100016279-A1 BICYCLIC DERIVATIVES FOR USE IN THE TREATMENT OF ANDROGEN RECEPTOR ASSOCIATED CONDITIONS-155 ASTRAZENECA AB (SE) 2010-01-21 US disclosed
WO-2009081197-A1 BICYCLIC DERIVATIVES FOR USE IN THE TREATMENT OF ANDROGEN RECEPTOR ASSOCIATED CONDITIONS ASTRAZENECA AB (SE) 2009-07-02 WO disclosed
WO-2008077597-A1 1-AMINOMETHYL- L- PHENYL- CYCLOHEXANE DERIVATIVES AS DDP-IV INHIBITORS NOVARTIS AG (CH) 2008-07-03 WO disclosed
US-7294625-B2 Pyrazole compounds UBE INDUSTRIES, LTD. (JP) 2007-11-13 US disclosed
US-20060063934-A1 3-Pyridazonyl- or triazolopyridazinyl- 4-pyridinyl- or pyrimidinyl- pyrazoles, e.g., 4-(2-aminopyridin-4-yl)-3-phenyl-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazole; p38MAP kinase inhibitors, used to treat rheumatoid arthritis UBE INDUSTRIES, LTD. (JP) 2006-03-23 US disclosed
EP-1553096-A1 PYRAZOLE COMPOUNDS Ube Industries, Ltd. (JP) 2005-07-13 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12344615-B2 Substituted pyridines as ion channel modulators SCN1A, CACNA1A, SCN5A ALDH1A1 819/4885KDM4E 836/4885SMN1; SMN2 147/4885
US-12152035-B2 Androgen receptor binding molecule and use thereof AR, SHBG, FSHR ALDH1A1 2266/4885KDM4E 1913/4885SMN1; SMN2 4854/4885
US-20250115569-A1 SULFONAMIDE COMPOUNDS FOR THE TREATMENT OF NEUROLOGICAL CONDITIONS CACNA1A, CACNA1E, CACNA1S ALDH1A1 3306/4885KDM4E 2441/4885SMN1; SMN2 84/4885
US-20060063934-A1 3-Pyridazonyl- or triazolopyridazinyl- 4-pyridinyl- or pyrimidinyl- pyrazoles, e.g., 4-(2-aminopyridin-4-yl)-3-phenyl-1-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)-1H-pyrazole; p38MAP kinase inhibitors, used to treat rheumatoid arthritis CNKSR1, MAPK1, MAPK3 ALDH1A1 2425/4885KDM4E 1462/4885SMN1; SMN2 4443/4885
US-20250163068-A1 COMPOUNDS AND THEIR METHODS OF USE SCN1A, SCN3A, SCN1B ALDH1A1 916/4885KDM4E 2066/4885SMN1; SMN2 334/4885
US-20260116885-A1 ION CHANNEL MODULATORS SCN1B, SCN1A, CACNA1S ALDH1A1 1251/4885KDM4E 3535/4885SMN1; SMN2 204/4885
US-20100267699-A1 CHEMICAL COMPOUNDS - 643 AR, KLK3, ESRRA ALDH1A1 377/4885KDM4E 1039/4885SMN1; SMN2 4314/4885
US-20100016279-A1 BICYCLIC DERIVATIVES FOR USE IN THE TREATMENT OF ANDROGEN RECEPTOR ASSOCIATED CONDITIONS-155 AR, NR5A1, CYP17A1 ALDH1A1 806/4885KDM4E 3067/4885SMN1; SMN2 3399/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.