SCHEMBL7502145

SCHEMBL7502145

O=c1[nH]nc(/C=C\c2cccnc2)c2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.51
CYP11B2 P19099 1/20 0.51
CHEK1 O14757 2/20 0.50
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
MAPT P10636 4/20 0.45
ALDH1A1 P00352 3/20 0.45
CYP1A1 P04798 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP1B1 Q16678 1/20 0.45
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
CRHBP P24387 1/20 0.43
CRHR2 Q13324 1/20 0.43
KDM4E B2RXH2 3/20 0.43
JUN P05412 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7502157 1.00 CYP11B1 (0.51) CYP11B1CYP11B2CHEK1KMT2AMEN1
SCHEMBL29214135 0.85 ATM (0.51) CHEK1KMT2AMEN1NPC1RAB9A
SCHEMBL5693205 0.82 CHEK1 (0.62) CYP11B1CYP11B2CHEK1KMT2AMEN1
SCHEMBL5693202 0.82 CHEK1 (0.62) CYP11B1CYP11B2CHEK1KMT2AMEN1
SCHEMBL5752477 0.81 PADI4 (0.44) ALDH1A1PADI4SMN1; SMN2
SCHEMBL5752478 0.81 PADI4 (0.44) ALDH1A1PADI4SMN1; SMN2
SCHEMBL7505673 0.81 PADI4 (0.44) ALDH1A1PADI4SMN1; SMN2
SCHEMBL4829935 0.74 TDO2 (0.60) CYP11B1CYP11B2KMT2AMEN1NPC1
SCHEMBL4832042 0.74 TDO2 (0.60) CYP11B1CYP11B2KMT2AMEN1NPC1
SCHEMBL12764197 0.74 CHEK1 (0.62) CYP11B1CYP11B2CHEK1CDK1CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165085-A1 PHTHALAZINE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES Novartis AG (CH) 2002-01-02 EP disclosed
WO-2000059509-A1 PHTHALAZINE DERIVATIVES FOR TREATING INFLAMMATORY DISEASES NOVARTIS AG (CH) 2000-10-12 WO disclosed