SCHEMBL7505992

SCHEMBL7505992

CCCCOc1cccc(C(=O)OCCCl)c1N

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.55
HSD17B10 Q99714 2/20 0.55
TSHR P16473 6/20 0.54
TDP1 Q9NUW8 2/20 0.54
L3MBTL1 Q9Y468 2/20 0.54
KDM4E B2RXH2 1/20 0.49
POLB P06746 1/20 0.49
CYP3A4 P08684 4/20 0.49
MAPK1 P28482 3/20 0.49
TP53 P04637 1/20 0.49
LMNA P02545 3/20 0.48
SLC6A3 Q01959 2/20 0.47
MAPT P10636 2/20 0.47
MEN1 O00255 1/20 0.47
NR1I2 O75469 1/20 0.47
CHRM2 P08172 1/20 0.47
ADRA2A P08913 1/20 0.47
OPRK1 P41145 1/20 0.47
HTR2B P41595 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7504921 0.95 ALDH1A1 (0.56) ALDH1A1HSD17B10TSHRTDP1L3MBTL1
SCHEMBL5710554 0.84 SCN1A (0.62) ALDH1A1HSD17B10TSHRTDP1L3MBTL1
SCHEMBL26696240 0.83 MAPT (0.51) ALDH1A1HSD17B10TSHRTDP1L3MBTL1
SCHEMBL7497377 0.83 ALDH1A1 (0.58) ALDH1A1HSD17B10TSHRTDP1L3MBTL1
SCHEMBL25438784 0.80 KMT2A (0.54) ALDH1A1HSD17B10TSHRTDP1L3MBTL1
SCHEMBL15771473 0.78 ALDH1A1 (0.64) ALDH1A1HSD17B10TSHRTDP1L3MBTL1
SCHEMBL4040621 0.77 ALDH1A1 (0.77) ALDH1A1HSD17B10TSHRTDP1L3MBTL1
SCHEMBL975212 0.77 TSHR (0.77) ALDH1A1HSD17B10TSHRTDP1L3MBTL1
SCHEMBL31091519 0.76 ALDH1A1 (0.66) ALDH1A1HSD17B10TSHRTDP1L3MBTL1
SCHEMBL23748669 0.76 TSHR (0.66) ALDH1A1HSD17B10TSHRTDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1124788-A4 BIS(HALOETHYL)AMINOBENZENE DERIVATIVES SHIONOGI BIORES CORP (US) 2002-11-06 EP claimed
EP-1124788-A2 BIS(HALOETHYL)AMINOBENZENE DERIVATIVES Shionogi Bioresearch Corporation (US) 2001-08-22 EP claimed
WO-2000024361-A2 BIS(HALOETHYL)AMINOBENZENE DERIVATIVES SHIONOGI BIORESEARCH CORP. (US) 2000-05-04 WO claimed
EP-1124788-A4 BIS(HALOETHYL)AMINOBENZENE DERIVATIVES SHIONOGI BIORES CORP (US) 2002-11-06 EP disclosed
EP-1250326-A2 INDAZOLE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND THEIR USE FOR MEDIATING OR INHIBITING CELL PROLIFERATION AGOURON PHARMACEUTICALS, INC. (US) 2002-10-23 EP disclosed
EP-1124788-A2 BIS(HALOETHYL)AMINOBENZENE DERIVATIVES Shionogi Bioresearch Corporation (US) 2001-08-22 EP disclosed
WO-2001053268-A2 INDAZOLE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND THEIR USE FOR MEDIATING OR INHIBITING CELL PROLIFERATION AGOURON PHARMACEUTICALS, INC. (US) 2001-07-26 WO disclosed
WO-2000024361-A2 BIS(HALOETHYL)AMINOBENZENE DERIVATIVES SHIONOGI BIORESEARCH CORP. (US) 2000-05-04 WO disclosed