SCHEMBL5710554

SCHEMBL5710554

CCCCOc1cccc(C(=O)OCCN(CC)CC)c1N

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 7/20 0.62
SCN2A Q99250 7/20 0.62
SCN3A Q9NY46 7/20 0.62
CYP2D6 P10635 5/20 0.62
CYP1A2 P05177 4/20 0.62
TSHR P16473 5/20 0.61
HRH3 Q9Y5N1 4/20 0.61
KCNH2 Q12809 3/20 0.61
SLC6A2 P23975 1/20 0.61
SLC6A3 Q01959 1/20 0.61
HIF1A Q16665 1/20 0.61
RAD52 P43351 1/20 0.60
MAOA P21397 3/20 0.53
CYP3A4 P08684 2/20 0.53
CYP2C19 P33261 1/20 0.53
SIGMAR1 Q99720 1/20 0.53
ALDH1A1 P00352 3/20 0.51
HSD17B10 Q99714 2/20 0.51
HTR3A P46098 3/20 0.50
CHRM2 P08172 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7505992 0.84 ALDH1A1 (0.55) SCN1ASCN2ASCN3ACYP2D6CYP1A2
SCHEMBL11339945 0.84 ALDH1A1 (0.62) SCN1ASCN2ASCN3ACYP2D6CYP1A2
SCHEMBL27629621 0.83 SCN1A (0.58) SCN1ASCN2ASCN3ACYP2D6CYP1A2
Metabutoxycaine SCHEMBL25778 0.83 ALDH1A1 (0.58) SCN1ASCN2ASCN3ACYP2D6CYP1A2
Metabutoxycaine SCHEMBL1643491 0.82 RAD52 (0.58) SCN1ASCN2ASCN3ACYP2D6CYP1A2
Metabutoxycaine SCHEMBL30053144 0.82 RAD52 (0.58) SCN1ASCN2ASCN3ACYP2D6CYP1A2
Ambucaine SCHEMBL82280 0.81 SCN1A (0.91) SCN1ASCN2ASCN3ACYP2D6CYP1A2
SCHEMBL11401080 0.81 SCN1A (0.67) SCN1ASCN2ASCN3ACYP2D6CYP1A2
Ambucaine SCHEMBL1007224 0.81 CYP2D6 (0.88) SCN1ASCN2ASCN3ACYP2D6CYP1A2
SCHEMBL26696240 0.80 MAPT (0.51) CYP1A2TSHRSLC6A3CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111295369-B Carbonic acid adducts 炎症药物有限责任公司 2023-07-25 CN disclosed
EP-1725098-A2 BENZAMIDE AND BENZOATE ANTI-HIV COMPOUNDS Samaritan Pharmaceuticals, Inc. (US) 2006-11-29 EP disclosed
WO-2005089453-A2 BENZAMIDE AND BENZOATE ANTI-HIV COMPOUNDS SAMARITAN PHARMACEUTICALS, INC. (US) 2005-09-29 WO disclosed