SCHEMBL7510189

SCHEMBL7510189

CC(C)C[C@H](NC(=O)CCCc1ccccc1)C(=O)N(C)C#N

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.52
CTSB P07858 4/20 0.52
CTSL P07711 4/20 0.52
CTSS P25774 3/20 0.52
CTSK P43235 3/20 0.52
HPGD P15428 1/20 0.50
LMNA P02545 2/20 0.48
PKM P14618 1/20 0.48
CTSG P08311 1/20 0.45
CMA1 P23946 1/20 0.45
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
ALDH1A1 P00352 2/20 0.44
NPC1 O15118 1/20 0.44
MAPT P10636 1/20 0.44
ALOX15 P16050 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4268532 0.81 SMN1; SMN2 (0.63) SMN1; SMN2HPGDLMNAPKMCTSG
SCHEMBL21759695 0.81 SMN1; SMN2 (0.63) SMN1; SMN2HPGDLMNAPKMCTSG
SCHEMBL6183685 0.81 CTSL (0.63) SMN1; SMN2CTSBCTSLCTSSCTSK
SCHEMBL20877889 0.79 SMN1; SMN2 (0.60) SMN1; SMN2HPGDLMNAPKMCTSG
SCHEMBL26259892 0.79 SMN1; SMN2 (0.60) SMN1; SMN2HPGDLMNAPKMCTSG
SCHEMBL22392193 0.78 SMN1; SMN2 (0.59) SMN1; SMN2HPGDLMNAPKMCTSG
SCHEMBL6183072 0.78 CTSK (0.80) CTSBCTSLCTSSCTSK
SCHEMBL26709736 0.77 SMN1; SMN2 (0.54) SMN1; SMN2CTSBCTSLCTSSCTSK
SCHEMBL9595087 0.76 SMN1; SMN2 (0.60) SMN1; SMN2HPGDLMNAPKMCTSG
SCHEMBL6019894 0.76 CTSL (0.51) CTSBCTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161415-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-12 EP disclosed
WO-2000055126-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed