SCHEMBL7510249

SCHEMBL7510249

O=CN(O)C(CO)CS(=O)(=O)c1ccc(-c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.65
AURKA O14965 1/20 0.65
NTRK1 P04629 1/20 0.65
MET P08581 1/20 0.65
PIM1 P11309 1/20 0.65
FGFR1 P11362 1/20 0.65
PRKACA P17612 1/20 0.65
GRK5 P34947 1/20 0.65
MAP2K2 P36507 1/20 0.65
FLT3 P36888 1/20 0.65
MAPK8 P45983 1/20 0.65
MAPK9 P45984 1/20 0.65
CDK8 P49336 1/20 0.65
GSK3B P49841 1/20 0.65
CDK7 P50613 1/20 0.65
CDK9 P50750 1/20 0.65
RPS6KA3 P51812 1/20 0.65
LIMK1 P53667 1/20 0.65
CDK5 Q00535 1/20 0.65
MAP2K1 Q02750 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7676525 0.90 CHEK1 (0.62) CHEK1AURKANTRK1METPIM1
SCHEMBL7679568 0.88 CHEK1 (0.60) CHEK1AURKANTRK1METPIM1
SCHEMBL7673400 0.86 MMP2 (0.67) CHEK1AURKANTRK1METPIM1
SCHEMBL7676192 0.84 MMP9 (0.87) MMP9MMP2MMP1
SCHEMBL7670905 0.84 CHEK1 (0.66) CHEK1AURKANTRK1METPIM1
SCHEMBL7673781 0.83 MMP9 (0.57) CHEK1AURKANTRK1METPIM1
SCHEMBL7673930 0.83 MMP2 (0.57) CHEK1AURKANTRK1METPIM1
SCHEMBL7451229 0.81 CHEK1 (0.57) CHEK1AURKANTRK1METPIM1
SCHEMBL7506195 0.81 CHEK1 (0.57) CHEK1AURKANTRK1METPIM1
SCHEMBL7670885 0.80 MMP9 (0.63) CHEK1AURKANTRK1METPIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001930-B1 N-HYDROXYFORMAMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES ABBOTT LAB (US) 2002-12-04 EP disclosed