SCHEMBL7512110

SCHEMBL7512110

O[C@@H]([C@H](O)[C@@H](COCc1ccc(C(F)(F)F)cc1)OCc1ccc(C(F)(F)F)cc1)[C@@H](COCc1ccc(C(F)(F)F)cc1)OCc1ccc(C(F)(F)F)cc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.46
TACR1 P25103 3/20 0.42
KMT2A Q03164 1/20 0.41
MAOB P27338 6/20 0.40
CACNA1F O60840 1/20 0.38
CACNA1D Q01668 1/20 0.38
CACNA1S Q13698 1/20 0.38
CACNA1C Q13936 1/20 0.38
PTPN2 P17706 1/20 0.38
PTPN1 P18031 1/20 0.38
PTPN6 P29350 1/20 0.38
SCN1A P35498 1/20 0.38
SCN5A Q14524 1/20 0.38
SCN9A Q15858 1/20 0.38
CA1 P00915 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7993000 0.94 TACR1 (0.47) IDO1TACR1CACNA1FCACNA1DCACNA1S
SCHEMBL7975619 0.94 TACR1 (0.47) IDO1TACR1CACNA1FCACNA1DCACNA1S
SCHEMBL7992780 0.82 IDO1 (0.41) IDO1MAOBCA1
SCHEMBL7515243 0.79 PRMT5 (0.42) MAOBCA1
SCHEMBL7510889 0.79 KCNH2 (0.44) TACR1KMT2AMAOBCA1
SCHEMBL5742123 0.78 CA1 (0.56) TACR1KMT2ACA1
SCHEMBL7990123 0.78 ESR1 (0.39) IDO1KMT2ACA1ALDH1A1
SCHEMBL7509273 0.77 CA1 (0.47) TACR1KMT2ACA1
SCHEMBL7989889 0.77 CA1 (0.47) TACR1KMT2ACA1
SCHEMBL7989942 0.77 CA1 (0.47) TACR1KMT2ACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1175385-A1 D-MANNITOL DERIVATIVES AS HIV ASPARTYL PROTEASE INHIBITORS Pharmacor Inc. (CA) 2002-01-30 EP disclosed
US-6313177-B1 AS ANTIVIRAL AGENTS PHARMACOR INC. (CA) 2001-11-06 US disclosed
WO-2000066524-A1 D-MANNITOL DERIVATIVES AS HIV ASPARTYL PROTEASE INHIBITORS PHARMACOR INC. (CA) 2000-11-09 WO disclosed