SCHEMBL7512504

SCHEMBL7512504

CCOC(=O)C(Cc1ccc(N)cc1)Nc1cc(Cl)ncn1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 8/20 0.48
ITGA4 P13612 8/20 0.48
PPID Q08752 3/20 0.42
ELANE P08246 1/20 0.39
CPB2 Q96IY4 2/20 0.36
PPIB P23284 1/20 0.36
PPIA P62937 1/20 0.36
PPIG Q13427 1/20 0.36
TACR1 P25103 1/20 0.36
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
TP53 P04637 1/20 0.36
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5368101 0.85 ITGB1 (0.64) ITGB1ITGA4
SCHEMBL5906839 0.79 ITGB1 (0.52) ITGB1ITGA4
SCHEMBL5906645 0.79 ITGB1 (0.52) ITGB1ITGA4
SCHEMBL5906642 0.79 ITGB1 (0.52) ITGB1ITGA4
SCHEMBL5906776 0.78 ALOX5 (0.40) ITGB1ITGA4
SCHEMBL2059146 0.77 PPID (0.43) PPIDELANECPB2PPIBPPIA
SCHEMBL27646223 0.77 FAAH (0.44) JAK2JAK3TP53
SCHEMBL27646221 0.77 FAAH (0.44) JAK2JAK3TP53
SCHEMBL30142880 0.73 PPID (0.53) PPIDPPIBPPIAPPIGTACR1
SCHEMBL2059018 0.72 ITGB1 (0.47) ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002008206-A1 3-AMINO-2-(4-AMINOCARBONYLOXY)PHENYL-PROPIONIC ACID DERIVATIVES AS ALPHA-4- INTEGRIN INHIBITORS ELAN PHARMACEUTICALS, INC. (US) 2002-01-31 WO disclosed