SCHEMBL7513745

SCHEMBL7513745

Nc1cc(F)c(S)cc1C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.50
KDM4E B2RXH2 6/20 0.46
ALDH1A1 P00352 5/20 0.46
HPGD P15428 2/20 0.46
HSD17B10 Q99714 2/20 0.46
IDO1 P14902 1/20 0.46
KMT2A Q03164 4/20 0.44
GFER P55789 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
TDP1 Q9NUW8 4/20 0.42
MAPT P10636 3/20 0.42
MEN1 O00255 3/20 0.42
THRB P10828 2/20 0.42
RECQL P46063 2/20 0.42
USP2 O75604 1/20 0.42
POLB P06746 1/20 0.42
PKM P14618 1/20 0.42
APEX1 P27695 1/20 0.42
BLM P54132 1/20 0.42
MCL1 Q07820 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL222733 0.83 KEAP1 (0.57) KEAP1KDM4EALDH1A1HPGDHSD17B10
Nitrogen SCHEMBL28658127 0.79 KEAP1 (0.53) KEAP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL24746192 0.78 CFTR (0.43) ALDH1A1KMT2AMEN1POLBCFTR
SCHEMBL17774726 0.78 KEAP1 (0.52) KEAP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL21664323 0.77 KDM4E (0.51) KEAP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL24418014 0.77 IDO1 (0.50) KEAP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL994342 0.76 KDM4E (0.50) KEAP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL3530679 0.76 KEAP1 (0.50) KEAP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL406782 0.76 KEAP1 (0.50) KEAP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL6018094 0.76 KDM4E (0.50) KEAP1KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001087842-A1 SUBSTITUTED POLYCYCLIC ARYL AND HETEROARYL PYRIDONES USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE PHARMACIA CORPORATION (US) 2001-11-22 WO claimed