SCHEMBL7513825

SCHEMBL7513825

OC(Nc1ncccn1)C1CCCC1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.50
GAA P10253 2/20 0.50
ALDH1A1 P00352 5/20 0.45
NPSR1 Q6W5P4 1/20 0.45
MAPK1 P28482 1/20 0.39
LCK P06239 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
MAPT P10636 1/20 0.34
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
GRM5 P41594 1/20 0.32
CTSK P43235 1/20 0.32
HTT P42858 1/20 0.32
HSD17B10 Q99714 1/20 0.32
RCE1 Q9Y256 1/20 0.32
IDO1 P14902 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12076597 0.73 ALDH1A1 (0.49) KDM4EGAAALDH1A1NPSR1LCK
SCHEMBL9664034 0.69 KDM4E (0.41) KDM4EGAAALDH1A1NPSR1SMN1; SMN2
SCHEMBL6190784 0.69 KDM4E (0.95) KDM4EGAAALDH1A1MAPK1CTSK
SCHEMBL15954538 0.67 KDM4E (1.00) KDM4EGAAALDH1A1MAPK1CTSK
SCHEMBL7768908 0.67 KDM4E (1.00) KDM4EGAAALDH1A1MAPK1CTSK
SCHEMBL1905978 0.66 CYP2C19 (0.39) KDM4EALDH1A1MAPK1CYP2C19KMT2A
SCHEMBL15045666 0.66 ALDH1A1 (0.42) KDM4EGAAALDH1A1NPSR1MAPK1
Isaxonine SCHEMBL1270289 0.65 KCNH3 (0.43) KDM4EGAAALDH1A1MAPK1LCK
SCHEMBL12162873 0.64 KDM4E (0.87) KDM4EGAAALDH1A1MAPK1CTSK
SCHEMBL21742249 0.64 TP53 (0.50) KDM4EALDH1A1SMN1; SMN2MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165522-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES Krenitsky Pharmaceuticals, Inc. (US) 2002-01-02 EP disclosed
WO-2000059893-A1 NEUROTROPHIC THIO SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC. (US) 2000-10-12 WO disclosed