SCHEMBL7514141

SCHEMBL7514141

O=C(CBr)c1cc(Cl)ccc1[N+](=O)[O-]

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
TSHR P16473 1/20 0.51
MAPK1 P28482 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
POLB P06746 1/20 0.47
MAPT P10636 3/20 0.46
PLA2G1B P04054 1/20 0.46
ATG4B Q9Y4P1 1/20 0.46
GAA P10253 1/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
HPGD P15428 2/20 0.46
CYP2C19 P33261 2/20 0.46
PKM P14618 1/20 0.45
GSK3B P49841 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8137810 0.87 HPGD (0.56) ALDH1A1KMT2AMEN1TSHRMAPK1
SCHEMBL2450846 0.85 ALDH1A1 (0.58) ALDH1A1KMT2AMEN1TSHRMAPK1
SCHEMBL2079317 0.84 ALDH1A1 (0.54) ALDH1A1KMT2AMEN1TSHRMAPK1
SCHEMBL18788570 0.82 GSK3B (0.45) ALDH1A1KMT2AMEN1MAPK1MAPT
SCHEMBL2080107 0.81 ALDH1A1 (0.52) ALDH1A1KMT2ATSHRMAPK1SMN1; SMN2
SCHEMBL10715141 0.80 ALDH1A1 (0.50) ALDH1A1KMT2AMEN1TSHRMAPK1
SCHEMBL8138933 0.80 GSK3B (0.42) ALDH1A1KMT2AMEN1TSHRMAPK1
SCHEMBL40329 0.80 ALDH1A1 (0.59) ALDH1A1KMT2AMEN1TSHRMAPK1
SCHEMBL79163 0.80 DTYMK (0.62) ALDH1A1KMT2AMEN1TSHRMAPK1
Hydrochloric Acid SCHEMBL1138798 0.78 DTYMK (0.60) ALDH1A1KMT2AMEN1TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001934-B1 INDOLE COMPOUNDS AS COX-2 INHIBITORS PFIZER (US) 2002-11-27 EP disclosed
US-6300363-B1 USEFUL IN THE TREATMENT OR ALLEVIATION OF INFLAMMATION AND OTHER INFLAMMATION ASSOCIATED DISORDERS IN MAMMALS PFIZER INC. 2001-10-09 US disclosed
EP-1001934-A1 INDOLE COMPOUNDS AS COX-2 INHIBITORS PFIZER PHARMACEUTICALS INC. (JP) 2000-05-24 EP disclosed
WO-1999005104-A1 INDOLE COMPOUNDS AS COX-2 INHIBITORS PFIZER PHARMACEUTICALS INC. (JP) 1999-02-04 WO disclosed