SCHEMBL7515374

SCHEMBL7515374

Cc1cc(C(F)(F)F)cc(C(=O)Nc2ccc3c(c2)CC(N2CCN(c4ccccn4)CC2)C3)c1-c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MTTP P55157 13/20 0.57
APOB P04114 10/20 0.57
SMO Q99835 10/20 0.52
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6200230 0.89 MTTP (0.72) MTTPAPOBSMO
SCHEMBL7505684 0.88 MTTP (0.59) MTTPAPOBSMO
SCHEMBL7561317 0.84 MTTP (0.78) MTTPAPOBSMO
SCHEMBL2990416 0.78 MTTP (0.67) MTTPAPOBSMO
SCHEMBL6199234 0.78 MTTP (0.75) MTTPAPOBSMO
SCHEMBL6201985 0.77 MTTP (0.72) MTTPAPOBSMO
SCHEMBL6198944 0.73 MTTP (0.78) MTTPAPOBSMO
SCHEMBL6195985 0.73 MTTP (0.78) MTTPAPOBSMO
SCHEMBL6201574 0.72 MTTP (1.00) MTTPAPOBSMO
SCHEMBL6198932 0.72 MTTP (1.00) MTTPAPOBSMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1259484-A1 CARBOXAMIDES USEFUL AS INHIBITORS OF MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN AND OF APOLIPOPROTEIN B SECRETION Novartis AG (CH) 2002-11-27 EP disclosed
WO-2001053260-A1 CARBOXAMIDES USEFUL AS INHIBITORS OF MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN AND OF APOLIPOPROTEIN B SECRETION NOVARTIS AG (CH) 2001-07-26 WO disclosed