SCHEMBL7515428

SCHEMBL7515428

COc1cc2c(Cc3ccncc3)n[nH]c(=O)c2cc1OC.COc1cc2c(cc1OC)C(=Cc1ccncc1)OC2=O

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ENPP1 P22413 3/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
PDE10A Q9Y233 1/20 0.45
ACHE P22303 4/20 0.42
AR P10275 1/20 0.40
MAOB P27338 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7515426 1.00 ENPP1 (0.47) ENPP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL6586097 0.82 ENPP1 (0.63) ENPP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL6586281 0.81 ACHE (0.54) CYP3A4CYP2C19ACHEMAOB
SCHEMBL6586280 0.81 ACHE (0.54) CYP3A4CYP2C19ACHEMAOB
SCHEMBL25548688 0.74 CYP2C9 (0.70) ENPP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL24000743 0.71 ENPP1 (0.74) ENPP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL8724175 0.70 KDM4E (0.60) CYP3A4CYP2C19ACHEMAOB
SCHEMBL8724172 0.70 KDM4E (0.60) CYP3A4CYP2C19ACHEMAOB
Hydrochloric Acid SCHEMBL30088793 0.70 ENPP1 (0.73) ENPP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL6589989 0.70 CYP11B1 (0.53) ENPP1CYP3A4CYP2C9TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1098886-A1 PHTHALAZINE DERIVATIVES AS PHOSPHODIESTERASE 4 INHIBITORS ZAMBON GROUP S.p.A. (IT) 2001-05-16 EP disclosed
WO-2000005219-A1 PHTHALAZINE DERIVATIVES AS PHOSPHODIESTERASE 4 INHIBITORS ZAMBON GROUP S.P.A. (IT) 2000-02-03 WO disclosed