SCHEMBL7517291

SCHEMBL7517291

CCOP(=O)(Cc1ccc(C(=O)N[C@@H](CC(C)C)C(=O)N[C@H]2CCO[C@H]2OC(C)=O)cc1)OCC

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 12/20 0.58
CAPNS1 P04632 2/20 0.57
CASP1 P29466 1/20 0.40
CASP3 P42574 1/20 0.40
CTSK P43235 6/20 0.40
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7513426 0.88 CAPN1 (0.55) CAPN1CAPNS1CASP1CASP3
SCHEMBL8810074 0.85 CAPN1 (0.66) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL8810052 0.85 CAPN1 (0.66) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL7517376 0.84 CAPN1 (0.65) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL8404221 0.84 CAPN1 (0.65) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL8404224 0.84 CAPN1 (0.65) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL7514155 0.78 CAPN1 (0.59) CAPN1CAPNS1CTSK
SCHEMBL27428998 0.78 CAPN1 (0.59) CAPN1CAPNS1CTSK
SCHEMBL27428996 0.78 CAPN1 (0.59) CAPN1CAPNS1CTSK
SCHEMBL8808938 0.76 CAPN1 (0.62) CAPN1CAPNS1CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP claimed
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP disclosed