SCHEMBL7517293

SCHEMBL7517293

Nc1nc[nH]c2cccc1-2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.41
GDA Q9Y2T3 2/20 0.36
MAP4K4 O95819 2/20 0.36
PARP1 P09874 1/20 0.35
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
TGFBR1 P36897 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
PIM1 P11309 1/20 0.33
PIM2 Q9P1W9 1/20 0.33
PNP P00491 2/20 0.33
PI4KA P42356 2/20 0.32
PI4K2B Q8TCG2 2/20 0.32
PI4K2A Q9BTU6 2/20 0.32
PI4KB Q9UBF8 2/20 0.32
LMNA P02545 1/20 0.32
DRD3 P35462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5255181 0.74 IDO1 (0.42) IDO1MAP4K4PARP1ALDH1A1POLB
SCHEMBL5733606 0.74 IDO1 (0.42) IDO1ALDH1A1POLBRXFP1ADRA2A
SCHEMBL3428780 0.70 IDO1 (0.46) IDO1GDAPI4KAPI4K2BPI4K2A
SCHEMBL21437991 0.68 HSD17B10 (0.44) IDO1PARP1ALDH1A1POLBRXFP1
SCHEMBL14674323 0.65 NUDT1 (0.39) MAP4K4ALDH1A1KDM4EGAAPI4KA
SCHEMBL1747899 0.65 KDM4A (0.37) IDO1GDAKDM4EGLAGAA
SCHEMBL87556 0.65 GDA (0.36) GDATGFBR1KDM4EGLAGAA
Hydrochloric Acid SCHEMBL3353320 0.64 KDM4A (0.36) IDO1GDAKDM4EPNPPI4KA
Hydrochloric Acid SCHEMBL29616692 0.64 GDA (0.35) GDAKDM4EPI4KAPI4K2BPI4K2A
Hydrochloric Acid SCHEMBL21683018 0.64 GDA (0.35) GDAKDM4EPI4KAPI4K2BPI4K2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2912019-A1 HETEROARYL INHIBITORS OF PDE4 Tetra Discovery Partners LLC (US) 2015-09-02 EP disclosed
WO-2014066659-A9 HETEROARYL INHIBITORS OF PDE4 TETRA DISCOVERY PARTNERS, LLC. (US) 2015-02-12 WO disclosed
WO-2014066659-A1 HETEROARYL INHIBITORS OF PDE4 TETRA DISCOVERY PARTNERS, LLC. (US) 2014-05-01 WO disclosed
EP-0643061-B1 Novel cephalosporin antibiotics and processes for preparation thereof LUCKY LTD (KR) 2002-01-30 EP disclosed
US-5541175-A Cephalosporin antibiotics LUCKY, LTD. (KR) 1996-07-30 US disclosed
EP-0643061-A1 Novel cephalosporin antibiotics and processes for preparation thereof LUCKY LTD. (KR) 1995-03-15 EP disclosed