SCHEMBL7518323

SCHEMBL7518323

O=C(N1Cc2cc3ccccc3c(S(=O)(=O)Cl)c2C1)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.36
ESR2 Q92731 5/20 0.36
CYP2D6 P10635 1/20 0.35
ABHD6 Q9BV23 3/20 0.33
HSP90AA1 P07900 2/20 0.32
HSP90AB1 P08238 2/20 0.32
HPGD P15428 1/20 0.32
PKM P14618 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PIK3CA P42336 1/20 0.31
SLC6A9 P48067 1/20 0.31
PTGDR Q13258 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7789796 0.81 ESR1 (0.38) ESR1ESR2ABHD6HSP90AA1HSP90AB1
SCHEMBL29972841 0.80 ESR1 (0.34) ESR1ESR2ABHD6
SCHEMBL7521223 0.79 HPGD (0.34) ESR1ESR2HSP90AA1HPGD
SCHEMBL7529328 0.76 CYP3A4 (0.46) ESR1ESR2ABHD6HPGD
SCHEMBL7786861 0.76 ESR1 (0.53) ESR1ESR2ABHD6HSP90AA1HSP90AB1
SCHEMBL7789910 0.74 ESR1 (0.43) ESR1ESR2ABHD6HSP90AA1HSP90AB1
SCHEMBL7462013 0.73 ESR1 (0.46) ESR1ESR2ABHD6PKMSMN1; SMN2
SCHEMBL7523701 0.72 POLB (0.32) ESR1ESR2PKMSLC6A9
SCHEMBL7526887 0.70 ALDH1A1 (0.34) ESR1ESR2HSP90AA1HPGDSMN1; SMN2
SCHEMBL7522643 0.70 ALDH1A1 (0.34) ESR1ESR2HPGDPKMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003747-A4 CARBAPENEMS WITH NAPHTHOSULTAM DERIVATIVE LINKED VIA METHYLENE MERCK & CO INC (US) 2002-11-06 EP disclosed
US-6251890-B1 TREATING OR PREVENTING BACTERIAL INFECTIONS IN MAMMALIAN PATIENTS MERCK & CO., INC. 2001-06-26 US disclosed
EP-1003747-A1 CARBAPENEMS WITH NAPHTHOSULTAM DERIVATIVE LINKED VIA METHYLENE Merck & Co., Inc. (US) 2000-05-31 EP disclosed
WO-1999009032-A1 CARBAPENEMS WITH NAPHTHOSULTAM DERIVATIVE LINKED VIA METHYLENE MERCK & CO., INC. (US) 1999-02-25 WO disclosed