SCHEMBL7518599

SCHEMBL7518599

Cc1ccc(S(=O)(=O)OCCOc2ccc(Nc3ncc(-c4ccccc4C#N)cn3)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 4/20 0.43
KDR P35968 4/20 0.43
SCN9A Q15858 3/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA9 Q16790 1/20 0.39
AVPR2 P30518 1/20 0.38
OXTR P30559 1/20 0.38
AVPR1A P37288 1/20 0.38
MAPT P10636 2/20 0.37
TP53 P04637 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
FFAR1 O14842 1/20 0.37
GRM5 P41594 1/20 0.37
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
PTK2 Q05397 1/20 0.36
CHEK1 O14757 2/20 0.35
AR P10275 1/20 0.35
S1PR1 P21453 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6033236 0.84 KDR (0.67) CDK1KDRALDH1A1
SCHEMBL6033199 0.78 CDK1 (0.54) CDK1KDRCA12CA1CA9
SCHEMBL7518604 0.74 IKBKB (0.49) MEN1KMT2A
SCHEMBL6033219 0.73 KDR (0.67) CDK1KDR
SCHEMBL9663522 0.73 ALDH1A1 (0.54) CA12CA1CA9MAPTCASP3
SCHEMBL12751681 0.72 ALDH1A1 (0.51) CA12CA1CA9MAPTALDH1A1
SCHEMBL6033867 0.72 KDR (0.48) CDK1KDRCA12CA1CA9
Acetonitrile SCHEMBL27788037 0.72 CA12 (0.50) CA12CA1CA9TP53SMN1; SMN2
SCHEMBL8069545 0.71 CA12 (0.63) CA12CA1CA9SMN1; SMN2CASP3
SCHEMBL1395593 0.70 CA12 (0.55) CA12CA1CA9TP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020147339-A1 5-cyano-2-aminopyrimidine derivatives CELLTECH R&D LIMITED (GB) 2002-10-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020147339-A1 5-cyano-2-aminopyrimidine derivatives FLT1, FGFR1, KDR CDK1 59/4885KDR 3/4885SCN9A 3640/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.