SCHEMBL7520231

SCHEMBL7520231

NNC(=O)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.70
MAPT P10636 2/20 0.68
CA12 O43570 1/20 0.58
CA1 P00915 1/20 0.58
CA2 P00918 1/20 0.58
CA9 Q16790 1/20 0.58
GPR35 Q9HC97 1/20 0.55
P2RX1 P51575 5/20 0.53
LMNA P02545 1/20 0.53
ACP1 P24666 1/20 0.51
EPHX2 P34913 1/20 0.50
IKBKE Q14164 1/20 0.49
P2RX4 Q99571 1/20 0.49
P2RX7 Q99572 1/20 0.49
TACR1 P25103 1/20 0.49
MEN1 O00255 1/20 0.49
HTT P42858 1/20 0.49
RAB9A P51151 1/20 0.49
KMT2A Q03164 1/20 0.49
KDR P35968 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2681462 0.88 MAPT (0.78) ALDH1A1MAPTCA12CA1CA2
SCHEMBL966454 0.82 ALDH1A1 (1.00) ALDH1A1MAPTCA12CA1CA2
Hydrochloric Acid SCHEMBL5124471 0.81 ALDH1A1 (0.97) ALDH1A1MAPTCA12CA1CA2
SCHEMBL7951394 0.81 MAPT (1.00) ALDH1A1MAPTCA12CA1CA2
SCHEMBL28854422 0.81 ALDH1A1 (0.51) ALDH1A1MAPTCA12CA1CA2
SCHEMBL7524681 0.81 EPHX2 (0.78) ALDH1A1MAPTCA12CA1CA2
SCHEMBL4488889 0.80 MAPT (0.61) MAPTCA12CA1CA2CA9
SCHEMBL7692960 0.79 GPR35 (0.74) MAPTGPR35P2RX1LMNAACP1
SCHEMBL11001590 0.79 EPHX2 (0.81) MAPTCA12CA1CA2CA9
SCHEMBL671986 0.78 MAPT (0.78) ALDH1A1MAPTCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173420-A2 HETEROCYCLIC COMPOUNDS HAVING ANTITUMOR ACTIVITY Novuspharma S.p.A. (IT) 2002-01-23 EP disclosed
WO-2000053581-A2 HETEROCYCLIC COMPOUNDS HAVING ANTITUMOR ACTIVITY NOVUSPHARMA S.P.A. (IT) 2000-09-14 WO disclosed