SCHEMBL7521779

SCHEMBL7521779

CC(OS(=O)(=O)Cc1ccccc1)N(C)C(=O)OC(C)(C)C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 1/20 0.43
MAPT P10636 1/20 0.41
ATM Q13315 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA7 P43166 1/20 0.40
CA14 Q9ULX7 1/20 0.40
NPSR1 Q6W5P4 3/20 0.39
AKT1 P31749 2/20 0.39
ALDH1A1 P00352 3/20 0.39
HSD17B10 Q99714 2/20 0.39
FPR1 P21462 1/20 0.39
STS P08842 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 2/20 0.38
HPGD P15428 2/20 0.38
XBP1 P17861 2/20 0.38
HTT P42858 2/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31072911 0.79 MMP13 (0.45) MMP13MAPTATMCA12CA1
SCHEMBL31072916 0.76 MMP13 (0.45) MMP13MAPTATMCA12CA1
SCHEMBL7521782 0.75 MMP13 (0.39) MMP13MAPTATMNPSR1ALDH1A1
SCHEMBL12050814 0.75 BCHE (0.53) ATMHPGDSLC6A4
SCHEMBL6634035 0.74 ATM (0.45) MAPTATMCA12CA1CA7
SCHEMBL2499502 0.73 POLB (0.47) MAPTNPSR1ALDH1A1L3MBTL1HPGD
SCHEMBL30878162 0.73 POLB (0.47) MAPTNPSR1ALDH1A1L3MBTL1HPGD
SCHEMBL30307663 0.73 POLB (0.47) MAPTNPSR1ALDH1A1L3MBTL1HPGD
SCHEMBL2189397 0.72 ATM (0.45) MMP13ATMNPSR1AKT1ALDH1A1
SCHEMBL1401042 0.71 MMP13 (0.46) MMP13MAPTATMALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1171127-A2 PHARMACEUTICAL COMPOSITIONS CONTAINING PYRIDINE OR PYRIMIDINE DERIVATIVES FOR INHIBITION OF CYTOKINE PRODUCTION AND SECRETION Targacept, Inc. (US) 2002-01-16 EP disclosed
WO-2000062767-A2 PHARMACEUTICAL COMPOSITIONS CONTAINING PYRIDINE OR PYRIMIDINE DERIVATES FOR INHIBITION OF CYTOKINE PRODUCTION AND SECRETION TARGACEPT, INC. (US) 2000-10-26 WO disclosed
EP-1042274-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE R.J. REYNOLDS TOBACCO COMPANY (US) 2000-10-11 EP disclosed
WO-2000023418-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE R.J. REYNOLDS TOBACCO COMPANY (US) 2000-04-27 WO disclosed