SCHEMBL752259

SCHEMBL752259

CCCCCO[C@@H](CO)C(CCCCC)OP(=O)(O)OCCN

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PLA2G2C Q5R387 1/20 0.46
PTPN1 P18031 1/20 0.39
PLA2G2D Q9UNK4 1/20 0.39
LPAR3 Q9UBY5 5/20 0.37
LPAR1 Q92633 4/20 0.37
SMPD1 P17405 3/20 0.37
LPAR2 Q9HBW0 2/20 0.36
LAP3 P28838 2/20 0.36
S1PR2 O95136 5/20 0.35
S1PR1 P21453 5/20 0.35
S1PR3 Q99500 5/20 0.35
S1PR4 O95977 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2311014 0.91 PLA2G2C (0.44) PLA2G2CPTPN1
SCHEMBL1963907 0.91 PLA2G2C (0.44) PLA2G2CPTPN1
SCHEMBL4444982 0.91 PLA2G2C (0.44) PLA2G2CPTPN1
SCHEMBL4435691 0.91 PLA2G2C (0.44) PLA2G2CPTPN1
SCHEMBL1965773 0.91 PLA2G2C (0.44) PLA2G2CPTPN1
SCHEMBL1964499 0.90 PLA2G2C (0.41) PLA2G2CPTPN1PLA2G2DLPAR3LPAR1
SCHEMBL1964225 0.90 PLA2G2C (0.41) PLA2G2CPTPN1PLA2G2DLPAR3LPAR1
SCHEMBL1964153 0.89 PLA2G2C (0.43) PLA2G2C
SCHEMBL1962712 0.89 PLA2G2C (0.43) PLA2G2C
SCHEMBL1964685 0.89 PLA2G2C (0.43) PLA2G2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0845981-B1 COMPOSITIONS COMPRISING CATIONIC AMPHIPHILES AND CO-LIPIDS FOR INTRACELLULAR DELIVERY OF THERAPEUTIC MOLECULES GENZYME CORP (US) 2002-09-25 EP claimed
EP-0845981-A1 COMPOSITIONS COMPRISING CATIONIC AMPHIPHILES AND CO-LIPIDS FOR INTRACELLULAR DELIVERY OF THERAPEUTIC MOLECULES GENZYME CORPORATION (US) 1998-06-10 EP claimed
WO-1997046223-A1 COMPOSITIONS COMPRISING CATIONIC AMPHIPHILES AND CO-LIPIDS FOR INTRACELLULAR DELIVERY OF THERAPEUTIC MOLECULES GENZYME CORPORATION (US) 1997-12-11 WO claimed
EP-4301341-A1 LOADING OF ALGINATE MICROSPHERES Board of Regents, The University of Texas System (US) 2024-01-10 EP disclosed
EP-3972566-A1 RADIOTHERAPEUTIC MICROSPHERES Board of Regents, The University of Texas System (US) 2022-03-30 EP disclosed
WO-2020237042-A1 RADIOTHERAPEUTIC MICROSPHERES PHILLIPS WILLIAM T (US) 2020-11-26 WO disclosed
WO-2020118271-A1 FIBRIN-TARGETED POLYMERIZED SHELL LIPID MICROBUBBLES NANOVALENT PHARMACEUTICALS, INC. (US) 2020-06-11 WO disclosed
EP-2909230-A1 STABILIZATION OF BIOMIMETIC MEMBRANES Danisco US Inc. (US) 2015-08-26 EP disclosed
WO-2014063097-A1 STABILIZATION OF BIOMIMETIC MEMBRANES DANISCO US INC. (US) 2014-04-24 WO disclosed
EP-2709590-A1 ENHANCED GROWTH INHIBITION OF OSTEOSARCOMA BY CYTOTOXIC POLYMERIZED LIPOSOMAL NANOPARTICLES TARGETING THE ALCAM CELL SURFACE RECEPTOR Nanovalent Pharmaceuticals, Inc. (US) 2014-03-26 EP disclosed
EP-2637649-A2 COMPOUNDS AND METHODS FOR TREATING PAIN Akron Molecules GmbH (AT) 2013-09-18 EP disclosed
EP-2430151-A2 MENIGOCOCCUS VACCINE CONTAINING LIPOOLIGOSACCHARIDE (LOS) FROM MODIFIED STRAINS OF L6 IMMUNOTYPE NEISSERIA MENINGITIDIS Sanofi Pasteur (FR) 2012-03-21 EP disclosed
EP-2429531-A2 USE OF LIPID CONJUGATES IN THE TREATMENT OF DISEASES ASSOCIATED WITH VASCULATURE Yissum Research Development Company of the Hebrew University of Jerusalem Ltd. (IL) 2012-03-21 EP disclosed
WO-2011149985-A1 POLYMERIZED SHELL LIPID MICROBUBBLES AND USES THEREOF NANOVALENT PHARMACEUTICALS, INC. (US) 2011-12-01 WO disclosed
WO-2010131116-A2 USE OF LIPID CONJUGATES IN THE TREATMENT OF DISEASES ASSOCIATED WITH VASCULATURE YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD. (IL) 2010-11-18 WO disclosed
WO-2010130898-A2 MENIGOCOCCUS VACCINE CONTAINING LIPOOLIGOSACCHARIDE (LOS) FROM MODIFIED STRAINS OF L6 IMMUNOTYPE NEISSERIA MENINGITIDIS SANOFI PASTEUR (FR) 2010-11-18 WO disclosed
WO-2010059963-A2 PREPARATION AND METHODOLOGY OF SILK FIBROIN NANOPARTICLES THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2010-05-27 WO disclosed
WO-2003101482-A2 LIPOSOME VACCINE FORMULATIONS FOR FIN-FISH GENESIS GROUP INC. (CA) 2003-12-11 WO disclosed
EP-0845981-A1 COMPOSITIONS COMPRISING CATIONIC AMPHIPHILES AND CO-LIPIDS FOR INTRACELLULAR DELIVERY OF THERAPEUTIC MOLECULES GENZYME CORPORATION (US) 1998-06-10 EP disclosed
WO-1997046223-A1 COMPOSITIONS COMPRISING CATIONIC AMPHIPHILES AND CO-LIPIDS FOR INTRACELLULAR DELIVERY OF THERAPEUTIC MOLECULES GENZYME CORPORATION (US) 1997-12-11 WO disclosed