SCHEMBL7524850

SCHEMBL7524850

O=C1C=C(Nc2cccc(Br)c2)CN1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.47
NCOA1 Q15788 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43
EGFR P00533 10/20 0.43
MAP2K1 Q02750 1/20 0.42
RAPGEF4 Q8WZA2 1/20 0.41
AURKA O14965 1/20 0.40
AURKB Q96GD4 1/20 0.40
INCENP Q9NQS7 1/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
LMNA P02545 1/20 0.40
ALOX15 P16050 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
AKT1 P31749 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7515459 0.73 IDO1 (0.43) IDO1NCOA1NCOA3EGFRMAP2K1
SCHEMBL29961547 0.72 RAPGEF4 (0.61) IDO1EGFRRAPGEF4MEN1LMNA
SCHEMBL29961149 0.72 RAPGEF4 (0.61) IDO1EGFRRAPGEF4MEN1LMNA
SCHEMBL1687027 0.72 RAPGEF4 (0.61) IDO1EGFRRAPGEF4MEN1LMNA
SCHEMBL18786726 0.71 MKNK1 (0.55)
SCHEMBL18786724 0.69 MKNK1 (0.34)
SCHEMBL7519427 0.68 GRM4 (0.44) MAP2K1RAPGEF4MEN1KMT2A
SCHEMBL7294506 0.68 PIM1 (0.41) RAPGEF4MEN1NPC1LMNARAB9A
SCHEMBL72905 0.67 MEN1 (0.68) EGFRRAPGEF4MEN1LMNAALOX15
SCHEMBL13602809 0.66 KMT2A (0.50) MEN1NPC1LMNAALOX15KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173420-A2 HETEROCYCLIC COMPOUNDS HAVING ANTITUMOR ACTIVITY Novuspharma S.p.A. (IT) 2002-01-23 EP disclosed
WO-2000053581-A2 HETEROCYCLIC COMPOUNDS HAVING ANTITUMOR ACTIVITY NOVUSPHARMA S.P.A. (IT) 2000-09-14 WO disclosed