SCHEMBL7515459

SCHEMBL7515459

O=C1C=C(Nc2cccc(Br)c2)CO1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.43
MAOB P27338 1/20 0.41
RAPGEF4 Q8WZA2 1/20 0.41
NCOA1 Q15788 1/20 0.40
NCOA3 Q9Y6Q9 1/20 0.40
EGFR P00533 4/20 0.39
AKT1 P31749 1/20 0.39
MAP2K1 Q02750 1/20 0.38
TDO2 P48775 1/20 0.38
ALDH1A1 P00352 1/20 0.37
EPAS1 Q99814 1/20 0.37
GAA P10253 1/20 0.36
CA1 P00915 1/20 0.36
MMP2 P08253 1/20 0.36
CA14 Q9ULX7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7528584 0.81 GRM5 (0.48) MAOBALDH1A1GAA
SCHEMBL7518230 0.80 KDM4E (0.40) MAOBRAPGEF4ALDH1A1GAACA1
SCHEMBL7517596 0.80 ALDH1A1 (0.54) EGFRALDH1A1CA1
SCHEMBL7520161 0.78 KIF11 (0.52) RAPGEF4ALDH1A1GAA
SCHEMBL7524850 0.73 IDO1 (0.47) IDO1RAPGEF4NCOA1NCOA3EGFR
SCHEMBL29961547 0.71 RAPGEF4 (0.61) IDO1RAPGEF4EGFRTDO2ALDH1A1
SCHEMBL1687027 0.71 RAPGEF4 (0.61) IDO1RAPGEF4EGFRTDO2ALDH1A1
SCHEMBL29961149 0.71 RAPGEF4 (0.61) IDO1RAPGEF4EGFRTDO2ALDH1A1
SCHEMBL7520380 0.70 MT-CO2 (0.51) IDO1ALDH1A1GAA
SCHEMBL7524238 0.70 RAPGEF4 (0.46) RAPGEF4ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173420-A2 HETEROCYCLIC COMPOUNDS HAVING ANTITUMOR ACTIVITY Novuspharma S.p.A. (IT) 2002-01-23 EP disclosed
WO-2000053581-A2 HETEROCYCLIC COMPOUNDS HAVING ANTITUMOR ACTIVITY NOVUSPHARMA S.P.A. (IT) 2000-09-14 WO disclosed