SCHEMBL7528839

SCHEMBL7528839

COc1ccc(N[C]=O)c(C)c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.53
RAB9A P51151 2/20 0.47
ADRA2A P08913 1/20 0.46
ADRA2C P18825 1/20 0.46
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
FFAR4 Q5NUL3 2/20 0.43
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA9 Q16790 2/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
NPC1 O15118 1/20 0.41
S1PR4 O95977 1/20 0.40
ALDH1A1 P00352 2/20 0.40
F10 P00742 1/20 0.40
P2RX7 Q99572 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5465233 0.85 GAA (0.44) GAAMEN1KMT2AS1PR4ALDH1A1
SCHEMBL2203557 0.81 ALDH1A1 (0.56) GAARAB9ACA12CA1CA2
SCHEMBL2095306 0.80 RAB9A (0.44) GAARAB9AMEN1KMT2ANPC1
SCHEMBL1758610 0.78 KMT2A (0.53) GAACA12CA1CA2CA9
SCHEMBL1188763 0.76 RAB9A (0.42) GAARAB9AMEN1KMT2ANPC1
SCHEMBL1356507 0.76 MEN1 (0.50) RAB9AFFAR4MEN1KMT2ANPC1
SCHEMBL2204875 0.76 GAA (0.59) GAARAB9AADRA2AADRA2CADRA1D
SCHEMBL11821170 0.75 GAA (0.58) GAARAB9AADRA2AADRA2CADRA1D
SCHEMBL2866545 0.75 GAA (0.58) GAARAB9AADRA2AADRA2CADRA1D
SCHEMBL4791618 0.75 GAA (0.58) GAARAB9AADRA2AADRA2CADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP claimed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US claimed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO claimed
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP disclosed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US disclosed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO disclosed