SCHEMBL7529207

SCHEMBL7529207

CCCC/C=C(\C(N)=O)S(=O)(=O)O.[NaH]

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.37
EP300 Q09472 1/20 0.36
FAAH O00519 3/20 0.36
SOAT1 P35610 2/20 0.35
TP53 P04637 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35
CNR1 P21554 1/20 0.33
KDM4E B2RXH2 2/20 0.33
TSHR P16473 1/20 0.32
PPARA Q07869 2/20 0.32
F7 P08709 1/20 0.32
F3 P13726 1/20 0.32
EPHX2 P34913 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8089344 0.98 GRIK1 (0.38) GRIK1EP300FAAHSOAT1TP53
SCHEMBL7534289 0.89 GRIK1 (0.33) GRIK1FAAH
SCHEMBL3687542 0.86 GRIK1 (0.34) GRIK1FAAHSOAT1TP53MEN1
SCHEMBL9515807 0.82 FAAH (0.32) FAAHSOAT1TP53MEN1CYP1A2
SCHEMBL10600654 0.81 EP300 (0.47) GRIK1EP300FAAHCYP1A2CYP2C19
SCHEMBL9505671 0.81 EP300 (0.47) GRIK1EP300FAAHCYP1A2CYP2C19
SCHEMBL999986 0.78 GRIK1 (0.31) GRIK1
SCHEMBL4473788 0.75 EP300 (0.42) GRIK1EP300FAAHSOAT1TP53
SCHEMBL4473785 0.75 EP300 (0.42) GRIK1EP300FAAHSOAT1TP53
SCHEMBL8815359 0.75 EP300 (0.34) GRIK1EP300TSHRPPARAF7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0812311-B1 HIGHLY POLYMERIZABLE N-VINYLCARBOXYLIC ACID AMIDE AND PRODUCTION PROCESS THEREOF SHOWA DENKO KK (JP) 2002-03-20 EP disclosed
EP-0473881-B1 Liquid absorption agent SHOWA DENKO KK (JP) 2001-11-07 EP disclosed
US-6166253-A Process for producing N-(1-alkoxyethyl)carboxylic amides SHOWA DENKO K.K. (JP) 2000-12-26 US disclosed
US-6153708-A HAVING AN N-1,3-BUTADIENYLCARBOXYLIC ACID AMIDE CONTENT OF 30 PPM OR LESS. SHOWA DENKO KABUSHIKI KAISHA (JP) 2000-11-28 US disclosed
US-6143836-A PRODUCING HOMOPOLYMER OR COPOLYMER OF N-VINYLCARBOXYLIC ACID AMIDE BY POLYMERIZING HIGHLY POLYMERIZABLE N-VINYLCARBOXYLIC ACID AMIDE HAVING N-1,3-BUTADIENYLCARBOXYLIC ACID AMIDE CONTENT OF 30 PPM OR LESS; USE AS THICKENER SHOWA DENKO KABUSHIKI KAISHA (JP) 2000-11-07 US disclosed
EP-0799820-B1 Process producing n-(1-alkoxyethyl)carboxylic amides SHOWA DENKO KK (JP) 2000-11-02 EP disclosed
US-6072084-A THERMAL CRACKING OR CATALYTIC CRACKING OF N-(1-ALKOXYETHYL) CARBOXYLIC ACID AMIDE OR ETHYLIDENEBISCARBOXYLIC ACID AMIDE SHOWA DENKO K.K. (JP) 2000-06-06 US disclosed
US-5892115-A PRETREATMENT BY THERMAL OR CATALYTIC CRACKING OF N-(1-ALKOXYETHYL)CARBOXYLIC AMIDE OR ETHYLIDENEBISCARBOXYLIC ACID AMIDE SHOWA DENKO KABUSHIKI KAISHA (JP) 1999-04-06 US disclosed
US-5852214-A Process for producing n-(1-alkoxyethyl) carboxylic amides SHOWA DENKO K.K. (JP) 1998-12-22 US disclosed
US-5789619-A USED AS COAGULANTS, LIQUID ABSORBENTS, THICKENERS SHOWA DENKO KABUSHIKI KAISHA (JP) 1998-08-04 US disclosed
US-5788950-A Method for the synthesis of mixed metal oxide powders SHOWA DENKO K.K. (JP) 1998-08-04 US disclosed
US-5744118-A MIXING ABSORBENT RESIN AND METAL SALTS, SWELLING AND GELATION, ADJUSTMENT OF PH, PYROLYSIS AND ROASTING SHOWA DENKO K.K. (JP) 1998-04-28 US disclosed
EP-0799820-A1 Process producing n-(1-alkoxyethyl)carboxylic amides SHOWA DENKO KABUSHIKI KAISHA (JP) 1997-10-08 EP disclosed
EP-0510246-B1 Use of fine particulate crosslinked type n-vinylamide resin microgel SHOWA DENKO KK (JP) 1996-09-25 EP disclosed
US-5407996-A Contacting with an aqueous solution of metal ion or metal oxide to form a gel; calcining SHOWA DENKO K.K. (JP) 1995-04-18 US disclosed
US-5338815-A Used in thickeners, dispersion stabilizers and lubricants SHOWA DENKO K.K. (JP) 1994-08-16 US disclosed
US-5300606-A Crosslinked N-vinylamide resin SHOWA DENKO K.K. (JP) 1994-04-05 US disclosed
US-5280095-A N-vinylcarboxylic acid amine resin SHOWA DENKO K.K. (JP) 1994-01-18 US disclosed
EP-0510246-A1 Use of fine particulate crosslinked type n-vinylamide resin microgel SHOWA DENKO KABUSHIKI KAISHA (JP) 1992-10-28 EP disclosed
EP-0473881-A1 Liquid absorption agent SHOWA DENKO KABUSHIKI KAISHA (JP) 1992-03-11 EP disclosed