SCHEMBL7529398

SCHEMBL7529398

CN(C)CC(Cc1c[nH]c2ccccc12)(NCc1cc2ccccc2o1)C(=O)O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 9/20 0.61
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
NPC1 O15118 1/20 0.44
POLB P06746 1/20 0.44
MAPT P10636 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HTR1A P08908 2/20 0.39
ADRA2A P08913 2/20 0.39
ADRA2B P18089 2/20 0.39
ADRA2C P18825 2/20 0.39
MAOA P21397 2/20 0.39
ADRA1D P25100 2/20 0.39
HTR1B P28222 2/20 0.39
HTR2A P28223 2/20 0.39
HTR2C P28335 2/20 0.39
CHRNB4 P30926 2/20 0.39
CHRNA3 P32297 2/20 0.39
HTR7 P34969 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7529387 1.00 TACR1 (0.61) TACR1MEN1KMT2ANPC1POLB
Hydrochloric Acid SCHEMBL7569288 0.99 TACR1 (0.60) TACR1MEN1KMT2ANPC1POLB
Hydrochloric Acid SCHEMBL7569286 0.99 TACR1 (0.60) TACR1MEN1KMT2ANPC1POLB
SCHEMBL7525917 0.88 TACR1 (0.77) TACR1
SCHEMBL7525927 0.88 TACR1 (0.77) TACR1
SCHEMBL7532240 0.88 TACR1 (0.77) TACR1
SCHEMBL7469433 0.79 TACR1 (0.69) TACR1
SCHEMBL13524867 0.79 TACR1 (0.55) TACR1MEN1KMT2ANPC1POLB
SCHEMBL13525369 0.79 TACR1 (0.55) TACR1MEN1KMT2ANPC1POLB
SCHEMBL7469438 0.78 CCKBR (0.49) TACR1MEN1KMT2ANPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244653-A1 NON PEPTIDE TACHYKININ RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2002-10-02 EP disclosed
WO-2001046176-A2 NON PEPTIDE TACHYKININ RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 2001-06-28 WO disclosed