SCHEMBL7530478

SCHEMBL7530478

O=C(/C=C/c1ccccc1)CC(=O)Cc1ccc(Cl)c(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HAO1 Q9UJM8 1/20 0.51
TBXA2R P21731 1/20 0.46
PTGER1 P34995 1/20 0.46
PTGER4 P35408 1/20 0.46
PTGFR P43088 1/20 0.46
PTGER3 P43115 1/20 0.46
PTGER2 P43116 1/20 0.46
PTGIR P43119 1/20 0.46
PTGDR Q13258 1/20 0.46
MAPT P10636 2/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
KCNH2 Q12809 1/20 0.45
GPR183 P32249 1/20 0.44
ALDH1A1 P00352 1/20 0.44
BACE1 P56817 3/20 0.44
GSK3B P49841 1/20 0.44
APP P05067 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL243735 0.77 HAO1 (0.75) HAO1MAPTKDM4EMEN1RAB9A
SCHEMBL7403121 0.76 SIGMAR1 (0.51) KMT2ASIGMAR1PIK3CAPDPK1
SCHEMBL3439644 0.75 HAO1 (0.84) HAO1MAPTKDM4EMEN1RAB9A
SCHEMBL316674 0.75 HAO1 (0.84) HAO1MAPTKDM4EMEN1RAB9A
SCHEMBL9113934 0.73 HAO1 (0.68) HAO1MAPTKDM4EMEN1RAB9A
SCHEMBL9113928 0.73 HAO1 (0.68) HAO1MAPTKDM4EMEN1RAB9A
SCHEMBL4625988 0.71 TRPV1 (0.47) TBXA2RPTGER1PTGER4PTGFRPTGER3
SCHEMBL23792517 0.71 TDP1 (0.59) MEN1KMT2APYGLSIGMAR1PDPK1
SCHEMBL3197944 0.71 BACE1 (0.80) BACE1PYGL
SCHEMBL3197932 0.71 BACE1 (0.80) BACE1PYGL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP disclosed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO disclosed