SCHEMBL7531979

SCHEMBL7531979

CNC(C)C(OC(=O)C(Cl)(Cl)COc1ccccc1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.40
CYP2D6 P10635 3/20 0.40
CYP2C19 P33261 3/20 0.40
MEN1 O00255 3/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP1A2 P05177 2/20 0.40
GAA P10253 1/20 0.40
ADRA1A P35348 4/20 0.40
CHRM2 P08172 1/20 0.40
RGS12 O14924 1/20 0.40
GLA P06280 1/20 0.40
PKM P14618 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
ALOX12 P18054 1/20 0.40
ADRA2C P18825 1/20 0.40
NFKB1 P19838 1/20 0.40
HTR2A P28223 1/20 0.40
THPO P40225 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ephedrine SCHEMBL8076172 0.80 ADRA1A (0.56) KMT2ACYP2D6CYP2C19MEN1CYP3A4
SCHEMBL14771681 0.77 CYP3A4 (0.46) KMT2ACYP2D6CYP2C19MEN1CYP3A4
SCHEMBL14771672 0.77 CYP3A4 (0.46) KMT2ACYP2D6CYP2C19MEN1CYP3A4
SCHEMBL14771667 0.72 ALDH1A1 (0.51) KMT2ACYP2D6CYP2C19MEN1CYP3A4
SCHEMBL4650189 0.72 ALDH1A1 (0.51) KMT2ACYP2D6CYP2C19MEN1CYP3A4
SCHEMBL14771663 0.72 ALDH1A1 (0.51) KMT2ACYP2D6CYP2C19MEN1CYP3A4
SCHEMBL14771654 0.72 TSHR (0.46) KMT2ACYP2D6CYP2C19MEN1CYP3A4
SCHEMBL11142451 0.72 TSHR (0.46) KMT2ACYP2D6CYP2C19MEN1CYP3A4
SCHEMBL2323888 0.71 TSHR (0.45) KMT2ACYP2D6CYP2C19MEN1CYP3A4
SCHEMBL28360980 0.70 CYP3A4 (0.51) KMT2ACYP2D6CYP2C19MEN1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0854846-A1 METHOD OF RESOLVING RACEMIC MIXTURES BASF AKTIENGESELLSCHAFT (DE) 1998-07-29 EP claimed
WO-1997011927-A1 METHOD OF RESOLVING RACEMIC MIXTURES BASF AKTIENGESELLSCHAFT (DE) 1997-04-03 WO claimed
EP-0854846-B1 METHOD OF RESOLVING RACEMIC MIXTURES BASF AG (DE) 2002-04-17 EP disclosed
US-6015903-A Method of resolving racemic mixtures BASF AKTIENGESELLSCHAFT (DE) 2000-01-18 US disclosed