SCHEMBL7532137

SCHEMBL7532137

COc1c(C(=O)N(C(C)C)C(C)C)[c]ccc1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.40
ALDH1A1 P00352 3/20 0.37
MAPT P10636 2/20 0.37
KDM4E B2RXH2 2/20 0.37
LMNA P02545 1/20 0.37
HPGD P15428 1/20 0.37
MCOLN3 Q8TDD5 1/20 0.37
TSHR P16473 1/20 0.37
PDE4B Q07343 4/20 0.36
PDE4A P27815 3/20 0.36
PDE4C Q08493 3/20 0.36
PDE4D Q08499 3/20 0.36
HTT P42858 2/20 0.34
MITF O75030 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
BACE1 P56817 2/20 0.33
FGFR1 P11362 1/20 0.33
SRC P12931 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7463231 0.82 NPSR1 (0.43) NPSR1ALDH1A1MAPTKDM4ELMNA
SCHEMBL2856090 0.79 IKBKB (0.45) ALDH1A1KDM4ELMNAHPGDPDE4B
SCHEMBL7823588 0.69 PDE4B (0.40) NPSR1ALDH1A1MAPTKDM4ETSHR
SCHEMBL7467767 0.66 MEN1 (0.41) NPSR1ALDH1A1MAPTKDM4ELMNA
SCHEMBL8011568 0.65 KMT2A (0.41) NPSR1ALDH1A1MAPTLMNAHPGD
SCHEMBL30268201 0.64 NPSR1 (0.66) NPSR1ALDH1A1MAPTKDM4ELMNA
SCHEMBL28039230 0.63 PDE4B (0.50) NPSR1ALDH1A1MAPTKDM4EPDE4B
SCHEMBL8131195 0.62 NPSR1 (0.41) NPSR1ALDH1A1MAPTKDM4ELMNA
SCHEMBL458409 0.62 NPSR1 (0.59) NPSR1ALDH1A1MAPTKDM4ELMNA
SCHEMBL12505385 0.62 BCAT2 (0.41) NPSR1ALDH1A1MAPTKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244617-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE Ortho-McNeil Pharmaceutical, Inc. (US) 2002-10-02 EP disclosed
WO-2001047875-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-07-05 WO disclosed