SCHEMBL7532982

SCHEMBL7532982

COC(=O)[C@H](Cc1ccccc1)N(C(=O)OC(C)(C)C)S(=O)(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 2/20 0.46
ITGB7 P26010 2/20 0.46
CA12 O43570 2/20 0.44
CA7 P43166 2/20 0.44
CA14 Q9ULX7 2/20 0.44
ATM Q13315 2/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
POLB P06746 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KLK5 Q9Y337 2/20 0.43
CA1 P00915 1/20 0.42
NPSR1 Q6W5P4 3/20 0.41
CTSS P25774 2/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSK P43235 1/20 0.40
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17137969 0.84 ITGA4 (0.50) ITGA4ITGB7CA12CA7CA14
SCHEMBL13163803 0.84 ITGA4 (0.50) ITGA4ITGB7CA12CA7CA14
SCHEMBL7609380 0.84 ITGA4 (0.50) ITGA4ITGB7CA12CA7CA14
SCHEMBL8724329 0.83 ITGA4 (0.49) ITGA4ITGB7CA12CA7CA14
SCHEMBL8724334 0.83 ITGA4 (0.49) ITGA4ITGB7CA12CA7CA14
SCHEMBL12600955 0.83 ITGA4 (0.49) ITGA4ITGB7CA12CA7CA14
SCHEMBL6442123 0.79 ITGA4 (0.46) ITGA4ITGB7CA12CA7CA14
SCHEMBL7299632 0.79 ITGA4 (0.46) ITGA4ITGB7CA12CA7CA14
SCHEMBL1937057 0.79 ABCB1 (0.46) ITGA4ITGB7ATMPOLBKLK5
SCHEMBL6795785 0.78 PTPRB (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0739338-B1 SERINE PROTEASE INHIBITORS: DERIVATIVES OF ISOTHIAZOLIDIN-3-ONE-1,1 DIOXIDE AND 3-OXO-1,2,5-THIADIAZOLIDINE-1,1-DIOXIDE UNIV WICHITA STATE (US) 2002-04-10 EP disclosed
US-5550139-A ANTIINFLAMMATORY AGENT, ANTITUMOR AGENT, ANTICARCINOGENIC AGENT THE WICHITA STATE UNIVERSITY (US) 1996-08-27 US disclosed