SCHEMBL7534102

SCHEMBL7534102

NC(=O)Oc1cccc2[nH]c(-c3cnccc3OCCN3CCNCC3)nc12

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.43
DHODH Q02127 1/20 0.43
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
GNRHR P30968 7/20 0.38
HTR1A P08908 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
DRD2 P14416 5/20 0.36
DRD3 P35462 5/20 0.36
PIM1 P11309 1/20 0.36
FLT3 P36888 1/20 0.36
PIM3 Q86V86 1/20 0.36
BRSK1 Q8TDC3 1/20 0.36
AURKB Q96GD4 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6587227 0.96 PARP1 (0.44) PARP1DHODHKDM4EALDH1A1TDP1
SCHEMBL6587192 0.93 PARP1 (0.50) PARP1DHODHKDM4EGNRHRHTR1A
SCHEMBL6583586 0.92 PARP1 (0.51) PARP1DHODHKDM4EALDH1A1GNRHR
SCHEMBL6583719 0.91 PARP1 (0.43) PARP1DHODHKDM4EALDH1A1GNRHR
SCHEMBL6590117 0.89 PARP1 (0.51) PARP1DHODHKDM4EALDH1A1PIM1
SCHEMBL6806003 0.89 PARP1 (0.56) PARP1DHODHPIM1FLT3PIM3
SCHEMBL6584782 0.88 AURKA (0.46) PARP1DHODHKDM4EALDH1A1TDP1
SCHEMBL6589815 0.88 PARP1 (0.52) PARP1DHODHKDM4EALDH1A1PIM1
SCHEMBL6587697 0.87 AURKB (0.44) PARP1DHODHKDM4EALDH1A1DRD3
SCHEMBL6799952 0.84 PARP1 (0.56) PARP1DHODHPIM1FLT3PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed