SCHEMBL7538602

SCHEMBL7538602

COc1cccc(OC)c1C(=O)Nc1nc(=O)[nH]cc1C[C@H](NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.47
SCN9A Q15858 2/20 0.46
ACE P12821 2/20 0.45
ITGA4 P13612 2/20 0.43
ITGB7 P26010 2/20 0.43
CTSS P25774 2/20 0.43
CTSK P43235 2/20 0.43
CTSL P07711 2/20 0.43
MAPT P10636 2/20 0.41
TP53 P04637 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
ITGB2 P05107 1/20 0.39
ICAM1 P05362 1/20 0.39
ITGAL P20701 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
PTPN1 P18031 1/20 0.39
CCKAR P32238 1/20 0.39
CCKBR P32239 1/20 0.39
ITGB3 P05106 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7538530 0.90 ITGB2 (0.48) ITGA4ITGB7MAPTTP53SMN1; SMN2
SCHEMBL7539039 0.89 ITGB2 (0.48) TACR1SCN9AACEITGA4CTSS
SCHEMBL7547460 0.86 ITGB2 (0.56) ITGA4ITGB7MAPTTP53SMN1; SMN2
SCHEMBL7544812 0.86 ITGB2 (0.56) ITGA4ITGB7MAPTTP53SMN1; SMN2
SCHEMBL6807195 0.86 KMT2A (0.47) ITGA4ITGB7ITGB2ICAM1ITGAL
SCHEMBL7540780 0.86 ITGB2 (0.45) MAPTSMN1; SMN2ITGB2ICAM1ITGAL
SCHEMBL6807437 0.86 ITGA4 (0.41) ACEITGA4ITGB7MAPTSMN1; SMN2
SCHEMBL7539842 0.85 ITGB2 (0.51) ITGA4ITGB7ITGB2ICAM1ITGAL
SCHEMBL7544261 0.85 ITGB2 (0.51) ITGA4ITGB7ITGB2ICAM1ITGAL
SCHEMBL7538428 0.85 ITGB2 (0.55) ITGA4ITGB7ITGB2ICAM1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1209147-A1 CARBOXYLIC ACID DERIVATIVES AND ADHESION MOLECULE INHIBITORS CONTAINING THE SAME AS THE ACTIVE INGREDIENT TORAY INDUSTRIES, INC. (JP) 2002-05-29 EP disclosed