Indole

Indole

SCHEMBL7539426

C=CCNCc1cccc2cc[nH]c12.c1ccc2[nH]ccc2c1

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 2/20 0.45
TRPA1 O75762 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
ITGB2 P05107 1/20 0.45
ICAM1 P05362 1/20 0.45
ITGAL P20701 1/20 0.45
CA4 P22748 1/20 0.45
CA6 P23280 1/20 0.45
ADK P55263 1/20 0.45
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
MC5R P33032 1/20 0.38
MC1R Q01726 1/20 0.38
BACE1 P56817 1/20 0.35
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
SLC6A3 Q01959 2/20 0.34
DRD4 P21917 1/20 0.34
ADORA2A P29274 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2259268 0.92 HTR2A (0.45) AHRHTR2AHTR2CBACE1SLC6A2
SCHEMBL4985160 0.73 PKM (0.47) AHRHTR2AHTR2CMC5RMC1R
SCHEMBL11478614 0.72 HTR2A (0.51) AHRHTR2AHTR2CBACE1ADORA2A
SCHEMBL10759141 0.72 AHR (0.46) AHRBACE1
Indole SCHEMBL7487754 0.71 AHR (0.57) AHRTRPA1CA1CA2ITGB2
SCHEMBL8590547 0.70 MC5R (0.53) CA2MC5RMC1R
Indole SCHEMBL5317626 0.70 AHR (0.61) AHRTRPA1CA1CA2ITGB2
Indole SCHEMBL6254730 0.70 AHR (0.65) AHRTRPA1CA1CA2ITGB2
Indole SCHEMBL3138428 0.70 AHR (0.65) AHRTRPA1CA1CA2ITGB2
Indole SCHEMBL26612366 0.70 AHR (0.65) AHRTRPA1CA1CA2ITGB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1250334-A2 AGENTS AND METHODS FOR THE TREATMENT OF PROLIFERATIVE DISEASES ELI LILLY AND COMPANY (US) 2002-10-23 EP disclosed
EP-1242420-A2 AGENTS AND METHODS FOR THE TREATMENT OF PROLIFERATIVE DISEASES ELI LILLY AND COMPANY (US) 2002-09-25 EP disclosed
WO-2001044235-A2 AGENTS AND METHODS FOR THE TREATMENT OF PROLIFERATIVE DISEASES ELI LILLY AND COMPANY (US) 2001-06-21 WO disclosed
WO-2001044247-A2 AGENTS AND METHODS FOR THE TREATMENT OF PROLIFERATIVE DISEASES ELI LILLY AND COMPANY (US) 2001-06-21 WO disclosed