SCHEMBL7541018

SCHEMBL7541018

COc1ccc(C(=O)NC(Cc2c[nH]c(=O)nc2NC(=O)c2c(OC)cccc2OC)C(=O)O)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.45
MMP9 P14780 1/20 0.44
HDAC3 O15379 8/20 0.43
HDAC1 Q13547 8/20 0.43
HDAC2 Q92769 8/20 0.43
NCOR2 Q9Y618 5/20 0.43
ITGB2 P05107 2/20 0.43
ICAM1 P05362 2/20 0.43
ITGAL P20701 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
ECE1 P42892 1/20 0.43
CA2 P00918 1/20 0.43
PTPN1 P18031 1/20 0.42
TACR1 P25103 1/20 0.42
PPARG P37231 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7545203 0.93 ITGB2 (0.43) HDAC3HDAC1HDAC2ITGB2ICAM1
SCHEMBL7542032 0.92 FPR2 (0.41) KMT2AMMP9HDAC3HDAC1HDAC2
SCHEMBL7538530 0.92 ITGB2 (0.48) KMT2AITGB2ICAM1ITGALMEN1
SCHEMBL7540043 0.91 TACR1 (0.46) KMT2AITGB2ICAM1ITGALPTPN1
SCHEMBL7545919 0.91 ITGB2 (0.49) KMT2AMMP9HDAC3HDAC1HDAC2
SCHEMBL7539705 0.90 ITGB1 (0.49) KMT2AMMP9ITGB2ICAM1ITGAL
SCHEMBL7549315 0.88 ITGB2 (0.42) KMT2AITGB2ICAM1ITGALTACR1
SCHEMBL7544812 0.88 ITGB2 (0.56) KMT2AITGB2ICAM1ITGALMEN1
SCHEMBL7540780 0.88 ITGB2 (0.45) KMT2AITGB2ICAM1ITGALMEN1
SCHEMBL7547460 0.88 ITGB2 (0.56) KMT2AITGB2ICAM1ITGALMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1209147-A1 CARBOXYLIC ACID DERIVATIVES AND ADHESION MOLECULE INHIBITORS CONTAINING THE SAME AS THE ACTIVE INGREDIENT TORAY INDUSTRIES, INC. (JP) 2002-05-29 EP disclosed