SCHEMBL7543780

SCHEMBL7543780

Cc1ccccc1N1CCN(S(=O)(=O)CC23CCC(CC2NC[C@@H](N)CCS(C)(=O)=O)C3(C)C)CC1

nearest known ligand 0.77

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OXTR P30559 5/20 0.77
AVPR2 P30518 2/20 0.77
AVPR1A P37288 2/20 0.77
CYP3A4 P08684 1/20 0.77
TSHR P16473 1/20 0.77
MEN1 O00255 2/20 0.76
KMT2A Q03164 2/20 0.76
BLM P54132 1/20 0.76
PMP22 Q01453 1/20 0.76
OPRK1 P41145 1/20 0.76
TMEM97 Q5BJF2 1/20 0.76
SIGMAR1 Q99720 1/20 0.76
AVPR1B P47901 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303364 0.87 OXTR (1.00) OXTRAVPR2AVPR1ACYP3A4TSHR
SCHEMBL17423280 0.87 OXTR (1.00) OXTRAVPR2AVPR1ACYP3A4TSHR
SCHEMBL29766904 0.87 OXTR (1.00) OXTRAVPR2AVPR1ACYP3A4TSHR
SCHEMBL14829136 0.87 OXTR (1.00) OXTRAVPR2AVPR1ACYP3A4TSHR
SCHEMBL7278360 0.87 OXTR (1.00) OXTRAVPR2AVPR1ACYP3A4TSHR
SCHEMBL12636892 0.87 OXTR (1.00) OXTRAVPR2AVPR1ACYP3A4TSHR
SCHEMBL17423276 0.87 OXTR (1.00) OXTRAVPR2AVPR1ACYP3A4TSHR
SCHEMBL26813473 0.87 OXTR (1.00) OXTRAVPR2AVPR1ACYP3A4TSHR
Hydrochloric Acid SCHEMBL30515732 0.86 MEN1 (1.00) OXTRAVPR2AVPR1ACYP3A4TSHR
Hydrochloric Acid SCHEMBL29371071 0.86 MEN1 (1.00) OXTRAVPR2AVPR1ACYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5648352-A STOPPING LABOR MERCK & CO., INC. (US) 1997-07-15 US disclosed
WO-1996012476-A1 WET GRANULATION FORMULATION FOR A PIPERAZINYLCAMPHORSULFONYL OXYTOCIN RECEPTOR ANTAGONIST MERCK & CO., INC. (US) 1996-05-02 WO disclosed
WO-1993006092-A1 PIPERAZINYL (SULFONYL)AMIDE DERIVATIVES OF CAMPHOR AS OXYTOCIN ANTAGONISTS MERCK & CO., INC. (US) 1993-04-01 WO disclosed
EP-0532097-A1 Piperazinyl(sulfon)amide derivatives of camphor as oxytocin antagonists MERCK & CO. INC. (US) 1993-03-17 EP disclosed