SCHEMBL7543969

SCHEMBL7543969

COC(=O)CCCN(C)c1ccc(Br)cc1C=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
KDM4E B2RXH2 4/20 0.40
HPGD P15428 1/20 0.40
ERN1 O75460 2/20 0.40
LTA4H P09960 1/20 0.39
KMT2A Q03164 3/20 0.37
CYP1A2 P05177 2/20 0.37
MEN1 O00255 2/20 0.37
ATM Q13315 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
TP53 P04637 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CASP3 P42574 1/20 0.36
TSHR P16473 1/20 0.36
MAPT P10636 2/20 0.36
POLB P06746 1/20 0.36
ALDH1A1 P00352 2/20 0.35
CYP2C19 P33261 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7541385 0.87 ALDH1A1 (0.44) PTGDR2KDM4EHPGDERN1LTA4H
SCHEMBL7541400 0.86 PTGDR2 (0.46) PTGDR2KDM4EERN1KMT2AMEN1
SCHEMBL5207046 0.86 PTGDR2 (0.39) PTGDR2KDM4EERN1KMT2ACYP1A2
SCHEMBL3458964 0.83 ALDH3A1 (0.42) EGFRPTGDR2KDM4EHPGDERN1
SCHEMBL5549984 0.83 PTGDR2 (0.45) PTGDR2KDM4EERN1KMT2AMEN1
SCHEMBL5551206 0.82 PTGDR2 (0.44) PTGDR2KDM4EERN1KMT2AMEN1
SCHEMBL3172718 0.81 PTGDR2 (0.35) EGFRPTGDR2KDM4EHPGDERN1
SCHEMBL24662160 0.80 HPGD (0.38) EGFRKDM4EHPGDLTA4HKMT2A
SCHEMBL6104478 0.79 ERN1 (0.41) EGFRPTGDR2KDM4EHPGDERN1
SCHEMBL3458699 0.78 BCHE (0.40) LTA4HKMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1211239-A1 PROCESS FOR THE PREPARATION OF 2,3-DIHYDROAZEPINE COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2002-06-05 EP disclosed