SCHEMBL7546647

SCHEMBL7546647

COc1ccc(-c2nc3ccccn3c2-c2ccc(S(C)(=O)=O)cc2)cc1OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.53
NR1I3 Q14994 2/20 0.48
KDM4E B2RXH2 3/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
GAA P10253 2/20 0.46
MAPT P10636 2/20 0.46
NPC1 O15118 1/20 0.45
TP53 P04637 1/20 0.45
PKM P14618 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HSD17B10 Q99714 1/20 0.45
KLK7 P49862 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
USP7 Q93009 1/20 0.44
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7222366 0.92 PTGS2 (0.53) PTGS2NR1I3KDM4EALDH1A1HPGD
SCHEMBL7216551 0.90 PTGS2 (0.52) PTGS2NR1I3
SCHEMBL7216393 0.90 PTGS2 (0.60) PTGS2NR1I3KDM4EALDH1A1GAA
SCHEMBL7221860 0.85 PTGS2 (0.71) PTGS2NR1I3KDM4EALDH1A1NPC1
SCHEMBL7218055 0.83 PTGS2 (0.64) PTGS2NR1I3NPC1RAB9AHDAC6
SCHEMBL7221442 0.83 ROCK2 (0.46) PTGS2KDM4EALDH1A1HPGDGAA
SCHEMBL7222378 0.83 PTGS2 (0.50) PTGS2NR1I3KDM4EALDH1A1HPGD
SCHEMBL7218017 0.81 PTGS2 (0.60) PTGS2NR1I3KDM4EALDH1A1GAA
SCHEMBL7221387 0.81 PTGS2 (0.60) PTGS2ALDH1A1
SCHEMBL7217081 0.80 PTGS2 (0.62) PTGS2NR1I3KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1104762-B1 SUBSTITUTED IMIDAZO[1,2A]AZINES AS SELECTIVE INHIBITORS OF COX-2 S A L V A T LAB SA (ES) 2002-09-18 EP claimed
EP-1104762-A1 SUBSTITUTED IMIDAZO 1,2A]AZINES AS SELECTIVE INHIBOTORS OF COX-2 LABORATORIOS S.A.L.V.A.T., S.A. (ES) 2001-06-06 EP claimed
EP-1104762-B1 SUBSTITUTED IMIDAZO[1,2A]AZINES AS SELECTIVE INHIBITORS OF COX-2 S A L V A T LAB SA (ES) 2002-09-18 EP disclosed
EP-1104762-A1 SUBSTITUTED IMIDAZO 1,2A]AZINES AS SELECTIVE INHIBOTORS OF COX-2 LABORATORIOS S.A.L.V.A.T., S.A. (ES) 2001-06-06 EP disclosed