SCHEMBL7547417

SCHEMBL7547417

O=C(O)c1ccc(N2CCNCC2)nc1.[KH]

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.52
HPGDS O60760 1/20 0.50
HDAC2 Q92769 6/20 0.48
HDAC3 O15379 4/20 0.48
SMO Q99835 1/20 0.48
ALDH1A1 P00352 2/20 0.48
ITGA2B P08514 1/20 0.47
OGA O60502 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
KMT2A Q03164 1/20 0.47
HDAC1 Q13547 4/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
LMNA P02545 1/20 0.47
HRH3 Q9Y5N1 1/20 0.46
PLD1 Q13393 1/20 0.46
USP2 O75604 1/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1896186 0.98 KCNH2 (0.53) KCNH2HPGDSHDAC2HDAC3SMO
Hydrochloric Acid SCHEMBL31552815 0.97 KCNH2 (0.52) KCNH2HPGDSHDAC2HDAC3SMO
SCHEMBL7550033 0.97 KCNH2 (0.52) KCNH2HPGDSHDAC2HDAC3SMO
SCHEMBL5202077 0.93 KCNH2 (0.49) KCNH2HPGDSHDAC2HDAC3SMO
SCHEMBL4935859 0.84 MAPT (0.51) KCNH2HPGDSHDAC2HDAC3ALDH1A1
SCHEMBL29524173 0.84 PARP1 (0.53) KCNH2HPGDSHDAC2HDAC3SMO
SCHEMBL2706925 0.84 PARP1 (0.53) KCNH2HPGDSHDAC2HDAC3SMO
SCHEMBL31352228 0.83 UBE2T (0.58) HPGDSSMOALDH1A1OGANPC1
SCHEMBL1989630 0.83 UBE2T (0.63) HPGDSSMOALDH1A1OGANPC1
SCHEMBL29784322 0.83 UBE2T (0.63) HPGDSSMOALDH1A1OGANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885886-B1 PYRIDINECARBOXAMIDE DERIVATIVES NISSHIN SEIFUN GROUP INC (JP) 2002-05-29 EP disclosed
US-5972943-A N-(NITRIC ACID,C14-18 ALKYL ESTER)-6-(1-(OPTIONALLY 4-SUBSTITUTED PIPERAZINYL)) PYRIDINE-3-CARBOXAMIDES; METHOD OF SYNTHESIS; ADMINISTERING TO TREAT CEREBRAL EDEMA; NO HYPOTENSIVE SIDE EFFECT NISSHIN FLOUR MILLING CO., LTD. (JP) 1999-10-26 US disclosed
EP-0885886-A1 NOVEL PYRIDINECARBOXAMIDE DERIVATIVES Nisshin Flour Milling Co., Ltd. (JP) 1998-12-23 EP disclosed