SCHEMBL7548170

SCHEMBL7548170

CCCn1nc(Cc2ccc(F)cc2)cc1C1CCN(N2CCC(c3cc(Cc4ccc(F)cc4)nn3C)CC2)CC1

nearest known ligand 0.41

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 19/20 0.41
PRCP P42785 1/20 0.41
KCNH2 Q12809 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7548174 0.88 PLAT (0.40) CCR5PRCP
SCHEMBL5763292 0.83 PLAT (0.42) CCR5PRCP
Hydrochloric Acid SCHEMBL7660201 0.82 PLAT (0.42) CCR5PRCP
SCHEMBL5763782 0.79 PLAT (0.44) CCR5PRCP
SCHEMBL5461506 0.73 CCR5 (0.46) CCR5PRCPKCNH2
Hydrochloric Acid SCHEMBL5764395 0.72 CCR5 (0.45) CCR5PRCPKCNH2
SCHEMBL5764492 0.71 CCR5 (0.47) CCR5PRCP
SCHEMBL5764913 0.70 PLAT (0.38) CCR5KCNH2
Hydrochloric Acid SCHEMBL5762051 0.70 CCR5 (0.47) CCR5
SCHEMBL27643633 0.70 CCR5 (0.49) CCR5PRCPKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1192133-A1 N-CYCLOPENTYL MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Merck & Co., Inc. (US) 2002-04-03 EP disclosed
WO-2000076972-A1 N-CYCLOPENTYL MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2000-12-21 WO disclosed