SCHEMBL7549839

SCHEMBL7549839

CCCc1c(Br)nc2ccc(Cl)cc2c1Br.CCCc1c(O)c2cc(Cl)ccc2[nH]c1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
MAPT P10636 1/20 0.51
KDM4E B2RXH2 7/20 0.48
HPGD P15428 4/20 0.48
SIRT1 Q96EB6 4/20 0.45
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42
HSD17B10 Q99714 4/20 0.41
GAA P10253 1/20 0.41
GSK3B P49841 1/20 0.41
TSHR P16473 1/20 0.40
ADORA1 P30542 1/20 0.38
TUBB4A P04350 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7120398 0.92 SIRT1 (0.46) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL7116460 0.84 ALDH1A1 (0.65) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL7551438 0.82 SIRT1 (0.38) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL7115559 0.82 KDM4E (0.44) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL7121362 0.80 SIRT1 (0.55) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL7117408 0.75 ALDH1A1 (0.65) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL7114815 0.75 ALDH1A1 (0.67) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL7120420 0.71 HSD17B10 (0.74) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL7121392 0.70 KDM4E (0.65) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL17505210 0.70 ALDH1A1 (0.65) ALDH1A1MEN1KMT2AMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244629-A2 QUINOLONE COMPOUNDS FOR USE IN TREATING VIRAL INFECTIONS GLAXO GROUP LIMITED (GB) 2002-10-02 EP disclosed
WO-2001046150-A2 QUINOLONE COMPOUNDS FOR USE IN TREATING VIRAL INFECTIONS GLAXO GROUP LIMITED (GB) 2001-06-28 WO disclosed