SCHEMBL7549908

SCHEMBL7549908

c1ccc2c(c1)c(-c1cncc(-c3ccsc3)c1)cn2CCN1CCCCCC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 1.00
FLT1 P17948 4/20 0.89
FLT4 P35916 4/20 0.89
FLT3 P36888 1/20 0.45
CYP2A6 P11509 1/20 0.43
HTR7 P34969 1/20 0.41
CNR1 P21554 2/20 0.40
CNR2 P34972 2/20 0.40
NFATC1 O95644 1/20 0.40
GSK3B P49841 1/20 0.40
DYRK1A Q13627 1/20 0.40
SMYD2 Q9NRG4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7556531 1.00 KDR (1.00) KDRFLT1FLT4FLT3CYP2A6
SCHEMBL7554703 0.94 KDR (1.00) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7506453 0.91 KDR (1.00) KDRFLT1FLT4CNR1CNR2
SCHEMBL7557243 0.87 KDR (0.77) KDRFLT1FLT4CYP2A6HTR7
SCHEMBL7551421 0.87 KDR (0.77) KDRFLT1FLT4CYP2A6HTR7
SCHEMBL7550153 0.87 KDR (0.77) KDRFLT1FLT4FLT3CNR1
SCHEMBL7555190 0.86 KDR (1.00) KDRFLT1FLT4CYP2A6NFATC1
SCHEMBL7546102 0.86 KDR (0.75) KDRFLT1FLT4FLT3CYP2A6
SCHEMBL7993940 0.85 KDR (0.74) KDRFLT1FLT4CYP2A6HTR7
SCHEMBL7555658 0.85 KDR (0.73) KDRFLT1FLT4FLT3CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147107-A4 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO INC (US) 2002-05-22 EP claimed
EP-1147107-A1 NOVEL ANGIOGENESIS INHIBITORS Merck & Co., Inc. (US) 2001-10-24 EP claimed
WO-2000043393-A1 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO., INC. (US) 2000-07-27 WO claimed
EP-1147107-A4 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO INC (US) 2002-05-22 EP disclosed
EP-1147107-A1 NOVEL ANGIOGENESIS INHIBITORS Merck & Co., Inc. (US) 2001-10-24 EP disclosed
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed
WO-2000043393-A1 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO., INC. (US) 2000-07-27 WO disclosed